Urb-597

Urb-597

SCHEMBL29371698

NC(=O)c1cccc(-c2cccc(OC(=O)NC3CCCCC3)c2)c1

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Full drug profile on Sugi Atlas →

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
FAAH O00519 4/20 1.00
TRPA1 O75762 1/20 1.00
EPHX2 P34913 1/20 1.00
FAAH2 Q6GMR7 1/20 1.00
MGLL Q99685 1/20 1.00
HDAC6 Q9UBN7 1/20 1.00

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Urb-597 SCHEMBL93842 1.00 FAAH (1.00) FAAHTRPA1EPHX2FAAH2MGLL
SCHEMBL14187855 0.99 FAAH (0.98) FAAHTRPA1EPHX2FAAH2MGLL
SCHEMBL17175654 0.96 FAAH (0.93) FAAHTRPA1EPHX2FAAH2MGLL
SCHEMBL4750537 0.92 FAAH (0.86) FAAHTRPA1EPHX2FAAH2MGLL
SCHEMBL10089400 0.92 FAAH (0.84) FAAHTRPA1EPHX2FAAH2MGLL
SCHEMBL14188106 0.90 FAAH (0.82) FAAHTRPA1EPHX2FAAH2MGLL
SCHEMBL16118260 0.90 FAAH (0.81) FAAHTRPA1EPHX2FAAH2MGLL
SCHEMBL14722820 0.90 FAAH (0.81) FAAHTRPA1EPHX2FAAH2MGLL
SCHEMBL17165898 0.89 FAAH (1.00) FAAHTRPA1EPHX2FAAH2MGLL
SCHEMBL18685448 0.89 FAAH (0.80) FAAHTRPA1EPHX2FAAH2MGLL

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 158 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20250360137-A1 ENHANCEMENT OF THE EFFICACY OF SEROTONERGIC PSYCHEDELIC DRUGS IN THE TREATMENT OR PREVENTION OF CERTAIN NEUROPSYCHIATRIC DISORDERS THROUGH INHIBITION OF TYPE-9 PHOSPHODIESTERASES FREEDOM BIOSCIENCES INC (US) 2025-11-27 US claimed
EP-4618980-A1 ENHANCEMENT OF THE EFFICACY OF SEROTONERGIC PSYCHEDELIC DRUGS IN THE TREATMENT OR PREVENTION OF CERTAIN NEUROPSYCHIATRIC DISORDERS THROUGH INHIBITION OF TYPE-9 PHOSPHODIESTERASES Freedom Biosciences, Inc. (US) 2025-09-24 EP claimed
EP-3762034-B1 A FATTY ACID AMIDE HYDROLASE (FAAHI) INHIBITOR FOR USE IN INHIBITING THE CELLULAR ACCUMULATION OF A SPHINGOLIPID IN A SUBJECT THAT HAS LYSOSOMAL STORAGE DISEASE OR DISORDER WYLDER NATION FOUND (US) 2025-08-27 EP claimed
EP-4583859-A2 COMPOSITIONS FOR PREVENTING TRANSITION FROM ACUTE TO CHRONIC PAIN The Regents of University of California (US) 2025-07-16 EP claimed
CN-119326745-A Application of URB597 in preparation of medicine for treating chronic traumatic encephalopathy 天津医科大学总医院 2025-01-21 CN claimed
WO-2024225481-A1 AGENT FOR IMPROVING THERAPEUTIC RESPONSIVENESS IN CANCER IMMUNOTHERAPY WITH PD-1 INHIBITOR OR PD-L1 INHIBITOR 国立大学法人京都大学 2024-10-31 WO claimed
US-20240252486-A1 ALGOSTATIC AGENTS FOR PREVENTING TRANSITION FROM ACUTE TO CHRONIC PAIN UNIV CALIFORNIA (US) 2024-08-01 US claimed
WO-2024107445-A1 ENHANCEMENT OF THE EFFICACY OF SEROTONERGIC PSYCHEDELIC DRUGS IN THE TREATMENT OR PREVENTION OF CERTAIN NEUROPSYCHIATRIC DISORDERS THROUGH INHIBITION OF TYPE-9 PHOSPHODIESTERASES FREEDOM BIOSCIENCES, INC. (US) 2024-05-23 WO claimed
WO-2024055006-A2 COMPOSITIONS FOR PREVENTING TRANSITION FROM ACUTE TO CHRONIC PAIN THE REGENTS OF THE UNIVERSITY OF CALIFORNIA (US) 2024-03-14 WO claimed
US-20230375561-A1 METHODS FOR IDENTIFICATION, STRATIFICATION, AND TREATMENT OF CNS DISEASES KADDURAH DAOUK RIMA F (US) 2023-11-23 US claimed
WO-2022204140-A1 ALGOSTATIC AGENTS FOR PREVENTING TRANSITION FROM ACUTE TO CHRONIC PAIN THE REGENTS OF THE UNIVERSITY OF CALIFORNIA (US) 2022-09-29 WO claimed
WO-2022081350-A2 METHODS FOR IDENTIFICATION, STRATIFICATION, AND TREATMENT OF CNS DISEASES DUKE UNIVERSITY (US) 2022-04-21 WO claimed
EP-4747247-A1 NOVEL FATTY ACID AMIDE HYDROLASE MODULATORS, COMPOSITIONS COMPRISING THE SAME AND USES THEREOF Apogee Pharmaceuticals, Inc. (CA) 2026-05-27 EP disclosed
EP-4048809-B1 SYSTEMS AND METHODS FOR PREDICTING THERAPEUTIC SENSITIVITY TEMPUS AI INC (US) 2026-05-27 EP disclosed
EP-3938345-B1 CHARGED ION CHANNEL BLOCKERS AND METHODS FOR USE NOCION THERAPEUTICS INC (US) 2026-05-06 EP disclosed
US-20260116859-A1 Charged Ion Channel Blockers and Methods for Use NOCION THERAPEUTICS INC (US) 2026-04-30 US disclosed
CN-114126617-A Piezoelectric agonists for preventing or reversing abnormal amyloid deposition 东芬兰大学 2022-03-01 CN disclosed
US-11253594-B2 Drug combinations for protecting against neuronal cell death UNIVERSITY OF PITTSBURGH-OF THE COMMONWEALTH SYSTEM OF HIGHER EDUCATION (US) 2022-02-22 US disclosed
US-20220041552-A1 CHARGED ION CHANNEL BLOCKERS AND METHODS FOR USE PRESIDENT AND FELLOWS OF HARVARD COLLEGE (US) 2022-02-10 US disclosed
US-11235112-B2 Inhalable dry powders PULMATRIX OPERATING COMPANY, INC. (US) 2022-02-01 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (5 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20250360137-A1 ENHANCEMENT OF THE EFFICACY OF SEROTONERGIC PSYCHEDELIC DRUGS IN THE TREATMENT OR PREVENTION OF CERTAIN NEUROPSYCHIATRIC DISORDERS THROUGH INHIBITION OF TYPE-9 PHOSPHODIESTERASES PDE9A, PDE3A, PDE2A FAAH 51/4885TRPA1 2709/4885EPHX2 528/4885
US-20220041552-A1 CHARGED ION CHANNEL BLOCKERS AND METHODS FOR USE TRPV1, TRPV2, TRPA1 FAAH 318/4885TRPA1 3/4885EPHX2 748/4885
US-11253594-B2 Drug combinations for protecting against neuronal cell death NLN, CASP3, BAX FAAH 1839/4885TRPA1 3242/4885EPHX2 2521/4885
US-20260116859-A1 Charged Ion Channel Blockers and Methods for Use OPRL1, TRPV1, SCN2B FAAH 913/4885TRPA1 13/4885EPHX2 870/4885
US-20230375561-A1 METHODS FOR IDENTIFICATION, STRATIFICATION, AND TREATMENT OF CNS DISEASES SLC25A20, CPT2, NDUFAB1 FAAH 69/4885TRPA1 4562/4885EPHX2 1139/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.