Calothrixin B

Calothrixin B

SCHEMBL29375353

O=C1c2[nH]c3ccccc3c2C(=O)c2cnc3ccccc3c21

nearest known ligand 0.45

Full drug profile on Sugi Atlas →

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CDK4 P11802 2/20 0.45
CCND1 P24385 2/20 0.45
TOP2A P11388 2/20 0.41
IDO1 P14902 1/20 0.39
ALDH1A1 P00352 5/20 0.39
KDM4E B2RXH2 4/20 0.39
HPGD P15428 4/20 0.39
HSD17B10 Q99714 4/20 0.39
MAPT P10636 3/20 0.39
LMNA P02545 3/20 0.39
MEN1 O00255 2/20 0.39
KMT2A Q03164 2/20 0.39
NPSR1 Q6W5P4 1/20 0.39
TUBB4A P04350 1/20 0.39
TUBB P07437 1/20 0.39
TUBA3C P0DPH7 1/20 0.39
TUBA1B P68363 1/20 0.39
TUBA4A P68366 1/20 0.39
TUBB4B P68371 1/20 0.39
TUBB3 Q13509 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Calothrixin B SCHEMBL5222737 1.00 CDK4 (0.45) CDK4CCND1TOP2AIDO1ALDH1A1
SCHEMBL1103721 0.79 MEN1 (0.44) IDO1ALDH1A1KDM4EMAPTMEN1
SCHEMBL21561768 0.79 ALDH1A1 (0.56) CDK4CCND1ALDH1A1KDM4EHPGD
SCHEMBL16895263 0.76 DNMT1 (0.46) IDO1ALDH1A1KDM4EMAPTLMNA
Benzocarbazoledione SCHEMBL22541347 0.76 MAOA (0.54) CDK4CCND1ALDH1A1KDM4EHPGD
SCHEMBL459050 0.73 KMT2A (0.44) IDO1ALDH1A1KDM4EMAPTLMNA
SCHEMBL29641696 0.73 KMT2A (0.44) IDO1ALDH1A1KDM4EMAPTLMNA
SCHEMBL22541429 0.72 CDC25B (0.44) CDK4CCND1TOP2AALDH1A1KDM4E
SCHEMBL6503650 0.72 MAOA (0.54) CDK4CCND1ALDH1A1KDM4EHPGD
SCHEMBL30673946 0.72 MAOA (0.54) CDK4CCND1ALDH1A1KDM4EHPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3947333-A4 INDOLE-YNONE MEDIATED BENZOANNULATION PROCESS FOR THE PREPARATION OF CARBAZOLES- CARBAZOMYCIN A, CALOTHRIXIN B AND STAUROSPORINONE Council of Scientific & Industrial Research (IN) 2022-12-28 EP disclosed
EP-3947333-A1 INDOLE-YNONE MEDIATED BENZOANNULATION PROCESS FOR THE PREPARATION OF CARBAZOLES- CARBAZOMYCIN A, CALOTHRIXIN B AND STAUROSPORINONE Council of Scientific & Industrial Research (IN) 2022-02-09 EP disclosed
EP-3947333-A1 INDOLE-YNONE MEDIATED BENZOANNULATION PROCESS FOR THE PREPARATION OF CARBAZOLES- CARBAZOMYCIN A, CALOTHRIXIN B AND STAUROSPORINONE Council of Scientific & Industrial Research (IN) 2022-02-09 EP disclosed