Reminertant

Reminertant

SCHEMBL29376784

COc1cccc(OC)c1-c1cc(C(=O)NC2(C(=O)O)C3CC4CC(C3)CC2C4)nn1-c1ccnc2cc(Cl)ccc12

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Full drug profile on Sugi Atlas →

Known targets — ChEMBL curated mechanism

NTSR1

The experimentally established mechanism targets of Reminertant. The predicted profile below is derived independently by chemical similarity — agreement is a validation signal, a miss is honest.

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
NTSR1 known ✓ P30989 9/20 1.00
NTSR2 O95665 2/20 1.00
FPR3 P25089 1/20 1.00
GPR183 P32249 1/20 1.00
SORT1 Q99523 1/20 1.00
OPRM1 P35372 1/20 0.65
OPRD1 P41143 1/20 0.65

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Reminertant SCHEMBL1650932 1.00 NTSR1 (1.00) NTSR1NTSR2FPR3GPR183SORT1
SCHEMBL19026903 0.93 NTSR1 (0.87) NTSR1NTSR2FPR3GPR183SORT1
SCHEMBL7556717 0.90 NTSR1 (0.81) NTSR1NTSR2FPR3GPR183SORT1
SCHEMBL8590399 0.89 NTSR1 (0.80) NTSR1NTSR2FPR3GPR183SORT1
SCHEMBL9078221 0.85 NTSR1 (0.75) NTSR1NTSR2FPR3GPR183SORT1
SCHEMBL17114634 0.85 NTSR1 (0.75) NTSR1NTSR2FPR3GPR183SORT1
SCHEMBL17114585 0.85 NTSR1 (0.75) NTSR1NTSR2FPR3GPR183SORT1
SCHEMBL17114586 0.85 NTSR1 (0.74) NTSR1NTSR2FPR3GPR183SORT1
SCHEMBL17114581 0.85 NTSR1 (0.74) NTSR1NTSR2FPR3GPR183SORT1
SCHEMBL8591222 0.84 NTSR1 (0.72) NTSR1NTSR2FPR3GPR183SORT1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 197 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2025111482-A1 COMPLEXING AGENT SALT FORMULATIONS OF PHARMACEUTICAL COMPOUNDS AT LOW STOICHIOMETRIC RATIOS BEXSON BIOMEDICAL, INC. (US) 2025-05-30 WO claimed
CN-119074732-A Application of NTSR1 inhibitor in treating chronic nasosinusitis 南京市中西医结合医院 2024-12-06 CN claimed
US-20260146036-A1 CRYSTALLINE FORMS RAQUALIA PHARMA INC. (JP) 2026-05-28 US disclosed
US-20260139031-A1 FUSION PROTEIN LEVICEPT LTD (GB) 2026-05-21 US disclosed
EP-4377309-B1 CRYSTALLINE FORMS RAQUALIA PHARMA INC (JP) 2026-05-20 EP disclosed
US-20260115194-A1 NEW TREATMENTS FOR PAIN SEVENLESS THERAPEUTICS LTD (GB) 2026-04-30 US disclosed
US-12605447-B2 Stable formulations for radionuclide complexes ITM SOLUCIN GMBH (DE) 2026-04-21 US disclosed
EP-4719596-A1 FUSION PROTEIN Levicept Limited (GB) 2026-04-08 EP disclosed
EP-4720104-A1 LOW AFFINITY P75 NEUROTROPHIC RECEPTOR EXTRACELLULAR DOMAIN FUSED TO A FC MOIETY AS NGF ANTAGONIST THERAPY OF PAIN Levicept Limited (GB) 2026-04-08 EP disclosed
EP-4712957-A2 ISOANDROGRAPHOLIDE ANALOGS AND METHOD FOR TREATMENT USING THE SAME Enveda Therapeutics, Inc. (US) 2026-03-25 EP disclosed
EP-4712967-A2 G-PROTEIN COUPLED RECEPTOR ANTAGONIST Enveda Therapeutics, Inc. (US) 2026-03-25 EP disclosed
US-20220110923-A1 ESTERS AND CARBAMATES AS MODULATORS OF SODIUM CHANNELS VERTEX PHARMACEUTICALS INCORPORATED 2022-04-14 US disclosed
WO-2022071484-A1 3-HYDROXYOXINDOLE DERIVATIVES AS CRHR2 ANTAGONIST RAQUALIA PHARMA INC. (JP) 2022-04-07 WO disclosed
EP-3976594-A1 A THERAPEUTIC APPROACH FOR TREATING NON-INFECTIOUS OCULAR IMMUNOINFLAMMATORY DISORDERS The Schepens Eye Research Institute, Inc. (US) 2022-04-06 EP disclosed
CN-114206849-A Therapeutic methods for treating non-infectious ocular immunoinflammatory disorders 斯格本斯眼科研究所有限公司 2022-03-18 CN disclosed
EP-3965751-A1 PARA-AMINOHIPPURIC ACID (PAH) AS A RENAL PROTECTIVE SUBSTANCE ITM Isotope Technologies Munich SE (DE) 2022-03-16 EP disclosed
CN-114126654-A Para-aminohippuric acid (PAH) as a kidney protective substance 同位素技术慕尼黑有限公司 2022-03-01 CN disclosed
US-20220047505-A1 Controlled Absorption Water-Soluble Pharmaceutically Active Organic Compound Formulation for Once-Daily Administration STI PHARMA, LLC (US) 2022-02-17 US disclosed
US-20220041684-A1 ENGINEERED PLATELETS FOR TARGETED DELIVERY OF A THERAPEUTIC AGENT JPV01 LTD. (GB) 2022-02-10 US disclosed
EP-3947434-A2 ENGINEERED PLATELETS FOR TARGETED DELIVERY OF A THERAPEUTIC AGENT JPV01 Ltd (GB) 2022-02-09 EP disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (5 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-12605447-B2 Stable formulations for radionuclide complexes EPOR, CD47, PRCP NTSR1 71/4885NTSR2 158/4885FPR3 1144/4885
US-20260146036-A1 CRYSTALLINE FORMS PRKCD, CCT8, CRYZ NTSR1 4572/4885NTSR2 4106/4885FPR3 4422/4885
US-20260115194-A1 NEW TREATMENTS FOR PAIN SOS1, OPRL1, SOS2 NTSR1 122/4885NTSR2 148/4885FPR3 715/4885
US-20220110923-A1 ESTERS AND CARBAMATES AS MODULATORS OF SODIUM CHANNELS SCN10A, CACNA1A, SCN3A NTSR1 1608/4885NTSR2 1121/4885FPR3 3631/4885
US-20260139031-A1 FUSION PROTEIN NTRK2, BDNF, NGFR NTSR1 37/4885NTSR2 39/4885FPR3 383/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.