SCHEMBL2938747

SCHEMBL2938747

O=C(O)CN1C(=O)C(Cc2ccccc2)NC12CCN(C(=O)c1ccc([N+](=O)[O-])cc1Cl)CC2

nearest known ligand 0.47

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
LMNA P02545 4/20 0.47
HTT P42858 3/20 0.47
SMN1; SMN2 Q16637 2/20 0.47
ALDH1A1 P00352 6/20 0.42
NPC1 O15118 1/20 0.39
RAB9A P51151 1/20 0.39
CYP2C9 P11712 1/20 0.39
CYP2C19 P33261 1/20 0.39
HTR2B P41595 1/20 0.39
MAPK14 Q16539 1/20 0.39
KMT2A Q03164 3/20 0.39
MAPT P10636 3/20 0.38
POLB P06746 2/20 0.38
MEN1 O00255 1/20 0.37
SLC6A9 P48067 1/20 0.37
SLC6A5 Q9Y345 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1801523 0.85 LMNA (0.45) LMNAHTTSMN1; SMN2ALDH1A1NPC1
SCHEMBL1805257 0.85 LMNA (0.45) LMNAHTTSMN1; SMN2ALDH1A1NPC1
SCHEMBL3999880 0.82 LMNA (0.49) LMNAHTTSMN1; SMN2ALDH1A1NPC1
SCHEMBL2942653 0.80 HPGD (0.42) LMNAHTTALDH1A1KMT2AMAPT
SCHEMBL4037859 0.80 L3MBTL1 (0.48) LMNAHTTSMN1; SMN2ALDH1A1CYP2C9
SCHEMBL4037858 0.80 L3MBTL1 (0.48) LMNAHTTSMN1; SMN2ALDH1A1CYP2C9
SCHEMBL2934172 0.79 CYP2C9 (0.53) LMNAHTTSMN1; SMN2ALDH1A1CYP2C9
SCHEMBL2942498 0.77 AVPR1A (0.53) LMNAALDH1A1CYP2C9KMT2AMEN1
SCHEMBL2943001 0.77 MEN1 (0.39) CYP2C19KMT2AMEN1
SCHEMBL2941843 0.77 CYP2C9 (0.45) HTTSMN1; SMN2ALDH1A1CYP2C9CYP2C19

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1730147-B1 SUBSTITUTED 1,4,8-TRIAZASPIRO[4,5]DECAN-2-ON COMPOUNDS FOR USE IN THE TREATMENT OF OBESITY GRUENENTHAL GMBH (DE) 2010-02-03 EP claimed