Cilostazol

Cilostazol

SCHEMBL29389547

O=C1CCc2cc(OCCCCc3nnnn3C3CCCCC3)ccc2N1

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Full drug profile on Sugi Atlas →

Known targets — ChEMBL curated mechanism

PDE3A

The experimentally established mechanism targets of Cilostazol. The predicted profile below is derived independently by chemical similarity — agreement is a validation signal, a miss is honest.

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PDE3A known ✓ Q14432 7/20 1.00
PDE3B Q13370 7/20 1.00
MEN1 O00255 1/20 1.00
ABCC4 O15439 1/20 1.00
CACNA1F O60840 1/20 1.00
ABCB11 O95342 1/20 1.00
ALDH1A1 P00352 1/20 1.00
LMNA P02545 1/20 1.00
CYP1A2 P05177 1/20 1.00
CYP3A4 P08684 1/20 1.00
ADORA3 P0DMS8 1/20 1.00
CYP2C9 P11712 1/20 1.00
TSHR P16473 1/20 1.00
MAPK1 P28482 1/20 1.00
THPO P40225 1/20 1.00
OPRK1 P41145 1/20 1.00
BLM P54132 1/20 1.00
PMP22 Q01453 1/20 1.00
CACNA1D Q01668 1/20 1.00
KMT2A Q03164 1/20 1.00

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Cilostazol SCHEMBL1818013 1.00 PDE3B (1.00) PDE3BPDE3AMEN1ABCC4CACNA1F
Cilostazol SCHEMBL16128 1.00 PDE3B (1.00) PDE3BPDE3AMEN1ABCC4CACNA1F
SCHEMBL7307973 0.97 PDE3B (0.94) PDE3BPDE3AMEN1ABCC4CACNA1F
Cilostazol SCHEMBL5798390 0.96 PDE3B (0.93) PDE3BPDE3AMEN1ABCC4CACNA1F
Cilostazol SCHEMBL5798394 0.96 PDE3B (0.92) PDE3BPDE3AMEN1ABCC4CACNA1F
SCHEMBL12116425 0.93 PDE3B (0.86) PDE3BPDE3AMEN1ABCC4CACNA1F
SCHEMBL30151140 0.91 PDE3B (0.83) PDE3BPDE3AMEN1ABCC4CACNA1F
SCHEMBL29701270 0.91 PDE3B (0.83) PDE3BPDE3AMEN1ABCC4CACNA1F
SCHEMBL30151170 0.91 PDE3B (0.83) PDE3BPDE3AMEN1ABCC4CACNA1F
SCHEMBL29701268 0.91 PDE3B (0.83) PDE3BPDE3AMEN1ABCC4CACNA1F

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 59 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2023205369-A1 COMBINATORIAL PHARMACOTHERAPY FOR THE RESTORATION OF NEURO-FUNCTION AND COMBINATORIAL PHARMACOLOGICAL COMPOSITION THEREFORE NEURO-INNOVATORS, LLC. (US) 2023-10-26 WO claimed
CN-109310688-B Medicine for preventing and/or treating dementia 国立研究开发法人国立循环器病研究中心 2023-09-01 CN claimed
CN-116829545-B Substituted pyrazolylpiperidine carboxylic acids 拜耳公司 2026-05-15 CN disclosed
US-20260102416-A1 COMPOSITION OF MATTER FOR TREATING AT A MEDICAL CONDITION AND METHODS OF USE AND MANUFACTURE THEREOF TLCO HOLDINGS INC. (US) 2026-04-16 US disclosed
US-12595247-B2 Substituted pyrazolo piperidine carboxylic acids BAYER AKTIENGESELLSCHAFT (DE) 2026-04-07 US disclosed
EP-4704983-A2 TREATMENT OF MEMORY LOSS WITH PHOSPHODIESTERASE INHIBITORS Cyrano Therapeutics, Inc. (US) 2026-03-11 EP disclosed
US-12569493-B2 Treatment of chemosensory dysfunction from a coronavirus infection Cyrano Therapeutics Inc. (US) 2026-03-10 US disclosed
US-20260041690-A1 Treatment of Memory Loss with Phosphodiesterase Inhibitors CYRANO THERAPEUTICS INC (US) 2026-02-12 US disclosed
US-20250290934-A1 METHODS AND COMPOSITIONS FOR DIAGNOSING AND TREATING LOSS AND/OR DISTORTION OF TASTE OR SMELL CYRANO THERAPEUTICS, INC. 2025-09-18 US disclosed
US-12329753-B2 Phosphodiesterase inhibitor treatment CYRANO THERAPEUTICS, INC. (US) 2025-06-17 US disclosed
US-12298316-B2 Methods and compositions for diagnosing and treating loss and/or distortion of taste or smell CYRANO THERAPEUTICS, INC. (US) 2025-05-13 US disclosed
US-20220241273-A1 USE OF SGC ACTIVATORS FOR THE TREATMENT OF OPHTHALMOLOGIC DISEASES BAYER AG (DE) 2022-08-04 US disclosed
CN-108883112-B Compounds, compositions and methods for cancer patient stratification and cancer treatment 拜耳医药股份公司 2022-07-26 CN disclosed
CN-114699528-A Compositions and methods for PDE3A or SLFN12 expressing cancers 布罗德研究所股份有限公司 2022-07-05 CN disclosed
WO-2022122917-A1 THE USE OF SGC ACTIVATORS FOR THE TREATMENT OF OPHTHALMOLOGIC DISEASES BAYER AKTIENGESELLSCHAFT (DE) 2022-06-16 WO disclosed
CN-114601837-A Compounds, compositions and methods for cancer patient stratification and cancer treatment 拜耳医药股份公司 2022-06-10 CN disclosed
US-20220178947-A1 METHODS AND COMPOSITIONS FOR DIAGNOSING AND TREATING LOSS AND/OR DISTORTION OF TASTE OR SMELL CYRANO THERAPEUTICS, INC. 2022-06-09 US disclosed
CN-112288775-B Multi-target shielding tracking method based on long-term and short-term prediction model 武汉大学 2022-04-15 CN disclosed
CN-108366947-B Compositions and methods for PDE3A or SLFN12 expressing cancers 布罗德研究所股份有限公司 2022-03-29 CN disclosed
CN-114051417-A Drug dissolution type stent 大塚医疗器械有限公司 2022-02-15 CN disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (5 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20260041690-A1 Treatment of Memory Loss with Phosphodiesterase Inhibitors PDE2A, PDE4A, PDE3A PDE3A 3/4885PDE3B 6/4885MEN1 2658/4885
US-20220241273-A1 USE OF SGC ACTIVATORS FOR THE TREATMENT OF OPHTHALMOLOGIC DISEASES PRKG1, PGC, PRKG2 PDE3A 5/4885PDE3B 10/4885MEN1 4767/4885
US-20260102416-A1 COMPOSITION OF MATTER FOR TREATING AT A MEDICAL CONDITION AND METHODS OF USE AND MANUFACTURE THEREOF PDE8B, MGLL, PDE3B PDE3A 9/4885PDE3B 3/4885MEN1 461/4885
US-12569493-B2 Treatment of chemosensory dysfunction from a coronavirus infection PDE2A, PDE5A, PDE3B PDE3A 5/4885PDE3B 3/4885MEN1 2962/4885
US-12595247-B2 Substituted pyrazolo piperidine carboxylic acids SSB, PDK4, FPR1 PDE3A 356/4885PDE3B 346/4885MEN1 3721/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.