Salmeterol

Salmeterol

SCHEMBL29397921

OCc1cc([C@@H](O)CNCCCCCCOCCCCc2ccccc2)ccc1O

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Full drug profile on Sugi Atlas →

Known targets — ChEMBL curated mechanism

ADRB2

The experimentally established mechanism targets of Salmeterol. The predicted profile below is derived independently by chemical similarity — agreement is a validation signal, a miss is honest.

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ADRB2 known ✓ P07550 19/20 1.00
ADRB1 P08588 18/20 1.00
ADRB3 P13945 17/20 1.00
KDM4E B2RXH2 2/20 1.00
MEN1 O00255 2/20 1.00
TP53 P04637 2/20 1.00
CYP3A4 P08684 2/20 1.00
MAPK1 P28482 2/20 1.00
KMT2A Q03164 2/20 1.00
HTR1A P08908 1/20 1.00
CHRM5 P08912 1/20 1.00
DRD2 P14416 1/20 1.00
ADRA2B P18089 1/20 1.00
DRD4 P21917 1/20 1.00
SLC6A2 P23975 1/20 1.00
FPR3 P25089 1/20 1.00
ADRA1D P25100 1/20 1.00
HTR1D P28221 1/20 1.00
HTR1B P28222 1/20 1.00
HTR2A P28223 1/20 1.00

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Salmeterol SCHEMBL29393289 1.00 ADRB2 (1.00) ADRB2ADRB1ADRB3KDM4EMEN1
Salmeterol SCHEMBL4767 1.00 ADRB2 (1.00) ADRB2ADRB1ADRB3KDM4EMEN1
Salmeterol SCHEMBL4768 1.00 ADRB2 (1.00) ADRB2ADRB1ADRB3KDM4EMEN1
Salmeterol SCHEMBL4452108 1.00 ADRB2 (1.00) ADRB2ADRB1ADRB3KDM4EMEN1
SCHEMBL4450046 1.00 ADRB2 (1.00) ADRB2ADRB1ADRB3KDM4EMEN1
Salmeterol SCHEMBL7176067 0.99 ADRB2 (0.98) ADRB2ADRB1ADRB3KDM4EMEN1
Salmeterol SCHEMBL28889602 0.99 ADRB2 (0.98) ADRB2ADRB1ADRB3KDM4EMEN1
Salmeterol SCHEMBL29266779 0.99 ADRB2 (0.98) ADRB2ADRB1ADRB3KDM4EMEN1
Salmeterol SCHEMBL6152211 0.98 ADRB2 (0.96) ADRB2ADRB1ADRB3KDM4EMEN1
SCHEMBL4454918 0.98 ADRB2 (0.96) ADRB2ADRB1ADRB3KDM4EMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 25 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-111057696-B Hydroxynitrile lyase mutant and application thereof in synthesis of (R) -salmeterol 华东理工大学 2022-11-11 CN claimed
EP-4676481-A1 COMBINATION OF BETA-2-ADRENERGIC RECEPTOR AGONISTS AND GLP-1 RECEPTOR AGONISTS FOR USE IN TREATING HYPERGLYCAEMIA Atrogi AB (SE) 2026-01-14 EP disclosed
EP-4665321-A1 COMBINATIONS OF BETA 2-ADRENERGIC RECEPTOR AGONISTS AND METFORMIN FOR USE IN TREATING OBESITY AND REDUCING BODY FAT Atrogi AB (SE) 2025-12-24 EP disclosed
EP-4651867-A1 BETA 2-ADRENERGIC RECEPTOR AGONISTS FOR TREATMENT OR PREVENTION OF MUSCLE WASTING Atrogi AB (SE) 2025-11-26 EP disclosed
US-20250262170-A1 COMBINATIONS OF BETA 2-ADRENERGIC RECEPTOR AGONISTS AND BETA 3-ADRENERGIC RECEPTOR AGONISTS, AND MEDICAL USES THEREOF ATROGI AB (SE) 2025-08-21 US disclosed
US-12370352-B2 Nasal and ophthalmic delivery of aqueous corticosteroid solutions CYDEX PHARMACEUTICALS, INC. (US) 2025-07-29 US disclosed
EP-4511014-A1 COMBINATIONS OF BETA 2-ADRENERGIC RECEPTOR AGONISTS AND BETA 3-ADRENERGIC RECEPTOR AGONISTS, AND MEDICAL USES THEREOF Atrogi AB (SE) 2025-02-26 EP disclosed
WO-2024184408-A1 COMBINATION OF BETA-2-ADRENERGIC RECEPTOR AGONISTS AND GLP-1 RECEPTOR AGONISTS FOR USE IN TREATING HYPERGLYCAEMIA ATROGI AB (SE) 2024-09-12 WO disclosed
WO-2024170727-A1 COMBINATIONS OF BETA 2-ADRENERGIC RECEPTOR AGONISTS AND METFORMIN FOR USE IN TREATING OBESITY AND REDUCING BODY FAT ATROGI AB (SE) 2024-08-22 WO disclosed
WO-2024153813-A1 BETA 2-ADRENERGIC RECEPTOR AGONISTS FOR TREATMENT OR PREVENTION OF MUSCLE WASTING ATROGI AB (SE) 2024-07-25 WO disclosed
WO-2023097697-A1 METHOD FOR SYNTHESIZING (1R)-1-(2,2-DIMETHYL-4H-1,3-BENZODIOXIN-6-YL)OXAZOLIDIN-2-ONE 广东莱佛士制药技术有限公司 2023-06-08 WO disclosed
US-20230149327-A1 Use of Salmeterol as an Anti-Coronaviral Agent NATIONAL INSTITUTES OF HEALTH (NIH), U.S. DEPT. OF HEALTH AND HUMAN SERVICES (DHHS), U.S. GOVERNMENT 2023-05-18 US disclosed
US-11590089-B2 Beta-2 selective adrenergic receptor agonists THE BOARD OF TRUSTEES OF THE LELAND STANFORD JUNIOR UNIVERSITY (US) 2023-02-28 US disclosed
WO-2023279315-A1 USE OF 2\"-O-RHAMNOSYL ICARISIDE II IN MUSCLE REPAIR AND REGENERATION 中国科学院深圳先进技术研究院 2023-01-12 WO disclosed
CN-111057696-B Hydroxynitrile lyase mutant and application thereof in synthesis of (R) -salmeterol 华东理工大学 2022-11-11 CN disclosed
CN-111057696-B Hydroxynitrile lyase mutant and application thereof in synthesis of (R) -salmeterol 华东理工大学 2022-11-11 CN disclosed
CN-111057696-B Hydroxynitrile lyase mutant and application thereof in synthesis of (R) -salmeterol 华东理工大学 2022-11-11 CN disclosed
US-20220339414-A1 NASAL AND OPHTHALMIC DELIVERY OF AQUEOUS CORTICOSTEROID SOLUTIONS CITIBANK, N.A., AS ADMINISTRATIVE AGENT 2022-10-27 US disclosed
US-11464862-B2 DPI formulation containing sulfoalkyl ether cyclodextrin CYDEX PHARMACEUTICALS, INC. (US) 2022-10-11 US disclosed
CN-114057713-A Method for synthesizing (R) -salmeterol intermediate 广东莱佛士制药技术有限公司 2022-02-18 CN disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (5 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-11590089-B2 Beta-2 selective adrenergic receptor agonists ADRB2, ADRB1, ADRA2C ADRB2 1/4885ADRB1 2/4885ADRB3 5/4885
US-20250262170-A1 COMBINATIONS OF BETA 2-ADRENERGIC RECEPTOR AGONISTS AND BETA 3-ADRENERGIC RECEPTOR AGONISTS, AND MEDICAL USES THEREOF ADRB2, ADRB3, ADRB1 ADRB2 1/4885ADRB1 3/4885ADRB3 2/4885
US-11464862-B2 DPI formulation containing sulfoalkyl ether cyclodextrin DSP, DSC1, SAE1 ADRB2 1196/4885ADRB1 1315/4885ADRB3 1548/4885
US-12370352-B2 Nasal and ophthalmic delivery of aqueous corticosteroid solutions CRH, HRH1, IL5 ADRB2 40/4885ADRB1 25/4885ADRB3 29/4885
US-20220339414-A1 NASAL AND OPHTHALMIC DELIVERY OF AQUEOUS CORTICOSTEROID SOLUTIONS CRH, HRH1, IL5 ADRB2 40/4885ADRB1 25/4885ADRB3 29/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.