SCHEMBL29399998

SCHEMBL29399998

CN(C)S(=O)(=O)c1cc(N2CCN(CCCCC(F)(F)F)CC2)ccc1C(=O)O

nearest known ligand 0.41

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
DRD2 P14416 9/20 0.41
DRD4 P21917 9/20 0.41
GAA P10253 2/20 0.40
MAPT P10636 2/20 0.40
KDM4E B2RXH2 1/20 0.40
ALDH1A1 P00352 1/20 0.40
HTR1A P08908 2/20 0.39
KCNH2 Q12809 2/20 0.39
DRD3 P35462 1/20 0.38
HTR7 P34969 2/20 0.36
HTR2A P28223 1/20 0.36
HTR2C P28335 1/20 0.36
SIGMAR1 Q99720 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29384773 0.80 ERAP1 (0.45) DRD2DRD4MAPTALDH1A1DRD3
SCHEMBL22499595 0.80 ERAP1 (0.45) DRD2DRD4MAPTALDH1A1DRD3
SCHEMBL29402230 0.72 GSTO1 (0.45) GAAMAPTALDH1A1
SCHEMBL29403481 0.72 GSTO1 (0.45) GAAMAPTALDH1A1
SCHEMBL29401680 0.72 GSTO1 (0.46) GAAMAPTALDH1A1
SCHEMBL29688026 0.66 HTR1A (0.49) DRD2DRD4GAAKDM4EHTR1A
SCHEMBL23060175 0.65 BID (0.40) GAAMAPTALDH1A1
SCHEMBL7240468 0.65 HTR7 (0.50) DRD2DRD4MAPTALDH1A1HTR1A
SCHEMBL10865646 0.65 HTR1A (0.48) DRD2DRD4GAAMAPTHTR1A
SCHEMBL10865051 0.64 DRD4 (0.48) DRD2DRD4GAAMAPTHTR1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-114174259-A Modulators of intracellular chloride concentration 意大利学院科技基金会 2022-03-11 CN claimed
CN-114174259-A Modulators of intracellular chloride concentration 意大利学院科技基金会 2022-03-11 CN disclosed