SCHEMBL294027

SCHEMBL294027

[O]S(=O)(=O)c1ccc2ccccc2c1

nearest known ligand 0.65

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
LMNA P02545 3/20 0.65
L3MBTL1 Q9Y468 1/20 0.59
F2 P00734 2/20 0.53
PRSS1 P07477 2/20 0.53
PRSS2 P07478 2/20 0.53
PRSS3 P35030 2/20 0.53
CA1 P00915 2/20 0.52
CA2 P00918 2/20 0.52
CA9 Q16790 1/20 0.52
MCOLN3 Q8TDD5 2/20 0.52
TSHR P16473 1/20 0.52
SMN1; SMN2 Q16637 1/20 0.50
PKM P14618 3/20 0.49
ATM Q13315 1/20 0.49
CYP19A1 P11511 1/20 0.49
PKLR P30613 1/20 0.46
MEN1 O00255 1/20 0.46
KMT2A Q03164 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8813894 0.93 LMNA (0.57) LMNAL3MBTL1F2PRSS1PRSS2
SCHEMBL1952494 0.83 LMNA (0.68) LMNAL3MBTL1F2PRSS1PRSS2
SCHEMBL8813715 0.83 ALDH1A1 (0.52) LMNAL3MBTL1TSHR
SCHEMBL2064679 0.81 L3MBTL1 (0.59) LMNAL3MBTL1F2PRSS1PRSS2
SCHEMBL193715 0.79 LMNA (0.63) LMNAL3MBTL1F2PRSS1PRSS2
SCHEMBL12234418 0.79 LMNA (0.63) LMNAL3MBTL1F2PRSS1PRSS2
SCHEMBL1588805 0.79 LMNA (0.63) LMNAL3MBTL1F2PRSS1PRSS2
SCHEMBL193716 0.79 LMNA (1.00) LMNAL3MBTL1F2PRSS1PRSS2
SCHEMBL2238091 0.79 LMNA (0.63) LMNAL3MBTL1F2PRSS1PRSS2
SCHEMBL6113091 0.79 LMNA (0.63) LMNAL3MBTL1F2PRSS1PRSS2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 936 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1847568-B1 THERMOSETTING RESIN COMPOSITION, THERMOSETTING-RESIN MOLDING MATERIAL, AND CURED OBJECT OBTAINED THEREFROM SUMITOMO BAKELITE CO (JP) 2015-05-20 EP claimed
US-6197972-B1 CHEMICAL INTERMEDIATES FOR ANTICHOLESTEROL AGENTS JANSSEN PHARMACEUTICA N.V. (BE) 2001-03-06 US claimed
US-5977112-A Process of making substituted benzofurans MERCK PATENT GESELLSCHAFT MIT BESCHRANKTER HAFTUNG (DE) 1999-11-02 US claimed
US-5753652-A Antiretroviral hydrazine derivatives NOVARTIS CORPORATION (US) 1998-05-19 US claimed
EP-0521827-B1 Pharmacological active hydrazin derivatives and process for their preparation CIBA GEIGY AG (CH) 1996-09-25 EP claimed
EP-0447171-B1 Polysulfate of cyclodextrin derivative and process for preparing the same TANABE SEIYAKU CO (JP) 1994-11-02 EP claimed
US-5248675-A Viricides for HIV TANABE SEIYAKU CO., LTD. 1993-09-28 US claimed
EP-0447171-A2 Polysulfate of cyclodextrin derivative and process for preparing the same TANABE SEIYAKU CO., LTD. (JP) 1991-09-18 EP claimed
US-20240238257-A1 SYNTHETIC METHODS FOR PREPARATION OF 4-(2-CHLORO-4-METHOXY-5-METHYLPHENYL)-N-[(1S)-2-CYCLOPROPYL-1-(3-FLUORO-4-METHYLPHENYL)ETHYL]-5-METHYL-N-PROP-2-YNYL-1,3-THIAZOL-2-AMINE SANOFI (FR) 2024-07-18 US disclosed
EP-4400492-A1 ACRIDINE COMPOUND OSAKA UNIVERSITY (JP) 2024-07-17 EP disclosed
US-20240208999-A1 HETEROCYCLIC COMPOUND OTSUKA PHARMACEUTICAL CO., LTD. (JP) 2024-06-27 US disclosed
CN-118103359-A Preparation method of eribulin derivative 江苏恒瑞医药股份有限公司 2024-05-28 CN disclosed
CN-112239407-B Diester compound having dimethylcyclobutane ring, method for producing the same, and method for producing dimethylcyclobutane compound derived from the same 信越化学工业株式会社 2024-05-28 CN disclosed
EP-4370507-A1 HYDROGENATED QUINOXALINES Otsuka Pharmaceutical Co., Ltd. (JP) 2024-05-22 EP disclosed
US-3966703-A Asymmetrical frisazo dyestuffs derived from diazotized 2,7-diamino-carbazole BAYER AKTIENGESELLSCHAFT (DT) 1976-06-29 US disclosed
US-3956334-A CHOLESTEROL AND TRIGLYCERIDE LOWERING ACTIVITY IN BLOOD MERCK PATENT GESELLSCHAFT MIT BESCHRANKTER HAFTUNG (DT) 1976-05-11 US disclosed
US-3951986-A Novel 2-propanol derivatives and preparation thereof SUMITOMO CHEMICAL COMPANY, LIMITED (JA) 1976-04-20 US disclosed
US-3948949-A ANTIPHOLISTIC MERCK PATENT GESELLSCHAFT MIT BESCHRANKTER (DT) 1976-04-06 US disclosed
US-3933840-A ANTIPHLOGISTIC MERCK PATENT GESELLSCHAFT MIT BESCHRANKTER HAFTUNG (DT) 1976-01-20 US disclosed
US-3932487-A HYPOTENSIVE MERCK PATENT GESELLSCHAFT MIT BESCHRANKTER HAFTUNG (DT) 1976-01-13 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20240238257-A1 SYNTHETIC METHODS FOR PREPARATION OF 4-(2-CHLORO-4-METHOXY-5-METHYLPHENYL)-N-[(1S)-2-CYCLOPROPYL-1-(3-FLUORO-4-METHYLPHENYL)ETHYL]-5-METHYL-N-PROP-2-YNYL-1,3-THIAZOL-2-AMINE CYP21A2, NR5A1, HSD3B1 LMNA 2463/4885L3MBTL1 4402/4885F2 3286/4885
US-20240208999-A1 HETEROCYCLIC COMPOUND AHR, PDGFRA, PDGFRB LMNA 3284/4885L3MBTL1 4662/4885F2 116/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.