SCHEMBL2940845

SCHEMBL2940845

O=C(O)CN1C(=O)C(Cc2ccccc2)NC12CCN(C(=O)COCc1ccccc1)CC2

nearest known ligand 0.47

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
GRM5 P41594 12/20 0.47
ALDH1A1 P00352 2/20 0.42
LMNA P02545 1/20 0.37
SMN1; SMN2 Q16637 1/20 0.37
RAB9A P51151 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1803072 0.86 GRM5 (0.48) GRM5ALDH1A1
SCHEMBL1803348 0.85 GRM5 (0.43) GRM5ALDH1A1
SCHEMBL2938912 0.84 CYP3A4 (0.42) ALDH1A1LMNASMN1; SMN2
SCHEMBL2934783 0.82 CCR5 (0.40) ALDH1A1LMNASMN1; SMN2
SCHEMBL2932813 0.82 MEN1 (0.43) ALDH1A1LMNASMN1; SMN2
SCHEMBL2942516 0.81 SMN1; SMN2 (0.48) ALDH1A1LMNASMN1; SMN2RAB9A
SCHEMBL1803451 0.81 ALDH1A1 (0.44) GRM5ALDH1A1
SCHEMBL2943556 0.81 LMNA (0.49) ALDH1A1LMNASMN1; SMN2
SCHEMBL2941205 0.80 MEN1 (0.44) ALDH1A1LMNASMN1; SMN2
SCHEMBL2941530 0.79 HPGD (0.43) ALDH1A1LMNASMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1730147-B1 SUBSTITUTED 1,4,8-TRIAZASPIRO[4,5]DECAN-2-ON COMPOUNDS FOR USE IN THE TREATMENT OF OBESITY GRUENENTHAL GMBH (DE) 2010-02-03 EP claimed