SCHEMBL29435779

SCHEMBL29435779

Cc1cc(N(C)C(=O)OC(C)(C)C)cnc1Br

nearest known ligand 0.38

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
BRD4 O60885 2/20 0.38
PAX8 Q06710 1/20 0.38
CREBBP Q92793 1/20 0.33
AAK1 Q2M2I8 1/20 0.33
SSTR4 P31391 1/20 0.32
F2 P00734 2/20 0.32
IRAK4 Q9NWZ3 1/20 0.32
USP30 Q70CQ3 1/20 0.32
ABL1 P00519 1/20 0.32
FGFR3 P22607 1/20 0.31
KDR P35968 1/20 0.31
BACE1 P56817 1/20 0.31
LIPE Q05469 1/20 0.31
ALDH1A1 P00352 1/20 0.31
KAT8 Q9H7Z6 2/20 0.31
KAT6A Q92794 1/20 0.30
KAT5 Q92993 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29435629 0.83 NOS3 (0.39) BRD4PAX8CREBBPF2IRAK4
SCHEMBL851068 0.80 BRD4 (0.39) BRD4PAX8CREBBPAAK1ABL1
SCHEMBL14084481 0.80 PAX8 (0.41) BRD4PAX8CREBBPAAK1SSTR4
SCHEMBL22583529 0.79 KDM4E (0.32) ALDH1A1
SCHEMBL31141817 0.78 BRD4 (0.36) BRD4PAX8USP30FGFR3KDR
SCHEMBL29435558 0.77 BRD4 (0.34) BRD4PAX8CREBBPLIPEALDH1A1
SCHEMBL29081667 0.77 PAX8 (0.44) BRD4PAX8CREBBPSSTR4LIPE
SCHEMBL13188227 0.77 RAB9A (0.39) BRD4PAX8USP30ALDH1A1
SCHEMBL29581626 0.77 RAB9A (0.39) BRD4PAX8USP30ALDH1A1
SCHEMBL30615320 0.77 PAX8 (0.44) BRD4PAX8CREBBPSSTR4LIPE

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20250276967-A1 HETEROCYCLIC COMPOUNDS AND THEIR USE FOR TREATMENT OF HELMINTHIC INFECTIONS AND DISEASES SIGNAL PHARMACEUTICALS, LLC 2025-09-04 US disclosed
US-12338235-B2 Heterocyclic compounds and their use for treatment of helminthic infections and diseases CELGENE CORPORATION (US) 2025-06-24 US disclosed
US-11505548-B2 Heterocyclic compounds and their use for treatment of helminthic infections and diseases CELGENE CORPORATION (US) 2022-11-22 US disclosed
EP-3959207-A1 HETEROCYCLIC COMPOUNDS AND THEIR USE FOR TREATMENT OF HELMINTHIC INFECTIONS AND DISEASES Celgene Corporation (US) 2022-03-02 EP disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (3 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20250276967-A1 HETEROCYCLIC COMPOUNDS AND THEIR USE FOR TREATMENT OF HELMINTHIC INFECTIONS AND DISEASES CYP8B1, HAX1, HRH4 BRD4 2590/4885PAX8 4566/4885CREBBP 4455/4885
US-11505548-B2 Heterocyclic compounds and their use for treatment of helminthic infections and diseases CYP8B1, HAX1, HRH4 BRD4 2590/4885PAX8 4566/4885CREBBP 4455/4885
US-12338235-B2 Heterocyclic compounds and their use for treatment of helminthic infections and diseases CYP8B1, HAX1, HRH4 BRD4 2590/4885PAX8 4566/4885CREBBP 4455/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.