SCHEMBL29435558

SCHEMBL29435558

Cc1cc(N(C)C(=O)OC(C)(C)C)cnc1N=C=S

nearest known ligand 0.34

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
BRD4 O60885 2/20 0.34
PAX8 Q06710 1/20 0.34
GABRA1 P14867 1/20 0.32
GABRG2 P18507 1/20 0.32
GABRB3 P28472 1/20 0.32
GABRA5 P31644 1/20 0.32
GABRA3 P34903 1/20 0.32
GABRA2 P47869 1/20 0.32
GABRA6 Q16445 1/20 0.32
LIPE Q05469 1/20 0.30
CREBBP Q92793 1/20 0.30
ALDH1A1 P00352 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22583253 0.85 CACNA1G (0.34) BRD4PAX8LIPEALDH1A1
SCHEMBL22583203 0.82
SCHEMBL29435779 0.77 BRD4 (0.38) BRD4PAX8LIPECREBBPALDH1A1
SCHEMBL29435629 0.77 NOS3 (0.39) BRD4PAX8LIPECREBBPALDH1A1
SCHEMBL22583230 0.75 ALDH1A1 (0.37) LIPEALDH1A1
SCHEMBL29435617 0.74 P2RX3 (0.31)
SCHEMBL22582915 0.74 P2RX3 (0.31)
SCHEMBL29435573 0.74 ALDH1A1 (0.32) PAX8ALDH1A1
SCHEMBL22583395 0.72 APLNR (0.36) BRD4PAX8GABRA1GABRG2GABRB3
SCHEMBL30400464 0.70 PAX8 (0.40) BRD4PAX8CREBBP

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20250276967-A1 HETEROCYCLIC COMPOUNDS AND THEIR USE FOR TREATMENT OF HELMINTHIC INFECTIONS AND DISEASES SIGNAL PHARMACEUTICALS, LLC 2025-09-04 US disclosed
US-12338235-B2 Heterocyclic compounds and their use for treatment of helminthic infections and diseases CELGENE CORPORATION (US) 2025-06-24 US disclosed
US-11505548-B2 Heterocyclic compounds and their use for treatment of helminthic infections and diseases CELGENE CORPORATION (US) 2022-11-22 US disclosed
EP-3959207-A1 HETEROCYCLIC COMPOUNDS AND THEIR USE FOR TREATMENT OF HELMINTHIC INFECTIONS AND DISEASES Celgene Corporation (US) 2022-03-02 EP disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (3 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20250276967-A1 HETEROCYCLIC COMPOUNDS AND THEIR USE FOR TREATMENT OF HELMINTHIC INFECTIONS AND DISEASES CYP8B1, HAX1, HRH4 BRD4 2590/4885PAX8 4566/4885GABRA1 2750/4885
US-11505548-B2 Heterocyclic compounds and their use for treatment of helminthic infections and diseases CYP8B1, HAX1, HRH4 BRD4 2590/4885PAX8 4566/4885GABRA1 2750/4885
US-12338235-B2 Heterocyclic compounds and their use for treatment of helminthic infections and diseases CYP8B1, HAX1, HRH4 BRD4 2590/4885PAX8 4566/4885GABRA1 2750/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.