SCHEMBL29453752

SCHEMBL29453752

CC(Br)c1ccc(F)cc1F

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CES2 O00748 2/20 0.43
CES1 P23141 2/20 0.43
IDO1 P14902 1/20 0.41
TDO2 P48775 1/20 0.41
ALDH1A1 P00352 1/20 0.39
PDE2A O00408 2/20 0.37
SLC6A2 P23975 2/20 0.36
MC4R P32245 1/20 0.36
CYP3A4 P08684 1/20 0.36
CYP2D6 P10635 1/20 0.36
SLC6A4 P31645 1/20 0.36
SLC6A3 Q01959 1/20 0.36
RECQL P46063 1/20 0.36
PSEN1 P49768 2/20 0.35
PSEN2 P49810 2/20 0.35
APH1B Q8WW43 2/20 0.35
NCSTN Q92542 2/20 0.35
APH1A Q96BI3 2/20 0.35
PSENEN Q9NZ42 2/20 0.35
HDAC6 Q9UBN7 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14774740 1.00 CES2 (0.43) CES2CES1IDO1TDO2ALDH1A1
SCHEMBL18242589 0.82 CES2 (0.47) CES2CES1IDO1TDO2ALDH1A1
SCHEMBL1601682 0.82 PSEN1 (0.46) CES2CES1ALDH1A1SLC6A4RECQL
SCHEMBL28395189 0.81 CES2 (0.46) CES2CES1IDO1TDO2ALDH1A1
SCHEMBL84105 0.81 CES2 (0.46) CES2CES1IDO1TDO2ALDH1A1
SCHEMBL27568024 0.80 APLNR (0.38) CES2CES1PSEN1PSEN2APH1B
SCHEMBL22728414 0.80 ACHE (0.33) CES2CES1ALDH1A1CYP2D6PSEN1
SCHEMBL18103172 0.80 TRPA1 (0.42) PDE2ASLC6A2APLNR
SCHEMBL31690066 0.80 APLNR (0.49) ALDH1A1PDE2AAPLNR
SCHEMBL15861423 0.80 APLNR (0.49) ALDH1A1PDE2AAPLNR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-4652162-A1 INHIBITORS OF MPTP NRG Therapeutics LTD (GB) 2025-11-26 EP disclosed
EP-4558224-A1 PYRROLES AND IMIDAZOLES AS BET PROTEIN INHIBITORS Tay Therapeutics Limited (GB) 2025-05-28 EP disclosed
WO-2024153946-A1 INHIBITORS OF MPTP NRG THERAPEUTICS LTD (GB) 2024-07-25 WO disclosed
WO-2024018423-A1 PYRROLES AND IMIDAZOLES AS BET PROTEIN INHIBITORS Tay Therapeutics Limited (GB) 2024-01-25 WO disclosed
EP-3976186-A1 COMPOUNDS, COMPOSITIONS, AND METHODS OF USE Sage Therapeutics, Inc. (US) 2022-04-06 EP disclosed