SCHEMBL29457486

SCHEMBL29457486

Cc1cccc(-c2ccc(C(C)C(N)=O)nc2)n1

nearest known ligand 0.44

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
CYP2A6 P11509 1/20 0.44
IRAK4 Q9NWZ3 2/20 0.44
TGFBR1 P36897 15/20 0.43
GRM5 P41594 1/20 0.41
CCR1 P32246 1/20 0.41
CCR8 P51685 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13728633 0.82 CYP2A6 (0.51) CYP2A6IRAK4TGFBR1GRM5CCR1
SCHEMBL29457060 0.78 PTGS2 (0.46)
SCHEMBL29457352 0.78 KMO (0.42)
SCHEMBL14593498 0.77 HTT (0.44) IRAK4GRM5CCR1CCR8
SCHEMBL17675612 0.74 PIM2 (0.45)
SCHEMBL1851645 0.74 ADRA2A (0.42) CCR1CCR8
SCHEMBL3421947 0.73 CYP2A6 (0.65) CYP2A6TGFBR1GRM5CCR1CCR8
SCHEMBL30146674 0.73 CYP2A6 (0.65) CYP2A6TGFBR1GRM5CCR1CCR8
SCHEMBL29457088 0.73 CYP1A2 (0.38)
SCHEMBL29457476 0.73 CHEK1 (0.48) CYP2A6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2022073904-A1 MRGX2 ANTAGONISTS GLAXOSMITHKLINE INTELLECTUAL PROPERTY DEVELOPMENT LIMITED (GB) 2022-04-14 WO disclosed