SCHEMBL29457352

SCHEMBL29457352

Cc1cccc(-c2ccc(C(C)C(N)=O)nc2)c1

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KMO O15229 2/20 0.42
MAP4K4 O95819 1/20 0.42
DHODH Q02127 1/20 0.42
ICMT O60725 2/20 0.41
WNT3A P56704 1/20 0.41
GRIN2B Q13224 1/20 0.41
TLR8 Q9NR97 2/20 0.40
EGLN1 Q9GZT9 1/20 0.40
HSD17B1 P14061 2/20 0.39
HSD17B2 P37059 2/20 0.39
PSEN1 P49768 1/20 0.39
PSEN2 P49810 1/20 0.39
APH1B Q8WW43 1/20 0.39
NCSTN Q92542 1/20 0.39
APH1A Q96BI3 1/20 0.39
PSENEN Q9NZ42 1/20 0.39
PARP1 P09874 2/20 0.39
AKR1C3 P42330 1/20 0.39
AKR1C2 P52895 1/20 0.39
MKNK1 Q9BUB5 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29457060 0.84 PTGS2 (0.46) MAP4K4PARP1MKNK1MKNK2
SCHEMBL20437913 0.81 MAP4K4 (0.42) MAP4K4WNT3AGRIN2BHSD17B1HSD17B2
SCHEMBL29457486 0.78 CYP2A6 (0.44)
SCHEMBL1851645 0.77 ADRA2A (0.42) PARP1
SCHEMBL29457476 0.73 CHEK1 (0.48) EGLN1
SCHEMBL13680500 0.72 KMO (0.57) KMOMAP4K4DHODHWNT3AGRIN2B
SCHEMBL17675612 0.71 PIM2 (0.45) DHODHWNT3A
SCHEMBL12349144 0.71 MAP4K4 (0.68) MAP4K4MKNK1MKNK2
SCHEMBL4402515 0.71 HSD17B1 (0.61) KMOMAP4K4EGLN1HSD17B1HSD17B2
SCHEMBL29457160 0.70 MKNK1 (0.48) PARP1MKNK1MKNK2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2022073904-A1 MRGX2 ANTAGONISTS GLAXOSMITHKLINE INTELLECTUAL PROPERTY DEVELOPMENT LIMITED (GB) 2022-04-14 WO disclosed