SCHEMBL2946541

SCHEMBL2946541

Cc1cc(N2CCS(=O)(=O)CC2)ccc1-c1nc2c(N)nc(N)nc2[nH]1

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CDK1 P06493 1/20 0.41
CDK2 P24941 1/20 0.41
DHFR P00374 4/20 0.34
PDGFRB P09619 2/20 0.34
PDGFRA P16234 1/20 0.34
ALDH1A1 P00352 1/20 0.34
KDM5B Q9UGL1 1/20 0.34
ADORA2A P29274 2/20 0.33
ADORA1 P30542 2/20 0.33
TGFBR1 P36897 1/20 0.33
ACVR1 Q04771 1/20 0.33
ALK Q9UM73 1/20 0.33
TNKS O95271 1/20 0.32
PARP1 P09874 1/20 0.32
TNKS2 Q9H2K2 1/20 0.32
PDE7A Q13946 2/20 0.32
PDE7B Q9NP56 1/20 0.32
KDM4E B2RXH2 1/20 0.32
FGFR1 P11362 1/20 0.31
KDR P35968 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2946549 0.90 CDK1 (0.32) CDK1CDK2DHFRADORA2AADORA1
SCHEMBL2951931 0.85 PRKDC (0.42) CDK1CDK2DHFRALDH1A1ADORA2A
SCHEMBL2953661 0.78 CDK1 (0.33) CDK1CDK2PDE7A
SCHEMBL3040608 0.74 F9 (0.34) ALDH1A1ADORA2AADORA1KDM4E
SCHEMBL2953664 0.73
SCHEMBL2952943 0.72 MAP2K7 (0.45) ALKPDE7APDE7B
SCHEMBL2946551 0.71 CDK1 (0.41) CDK1CDK2DHFRPDGFRBPDGFRA
SCHEMBL2946044 0.71 MAPT (0.43) CDK1CDK2DHFRALDH1A1ADORA2A
SCHEMBL2955281 0.70 CAMKK2 (0.45) ADORA2APARP1
SCHEMBL2946368 0.70 PRKDC (0.40) CDK1CDK2DHFRADORA2AADORA1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010111406-A2 COMPOUNDS AND THERAPEUTIC USES THEREOF MYRIAD PHARMACEUTICALS, INC. (US) 2010-09-30 WO claimed