SCHEMBL2946549

SCHEMBL2946549

Cc1cc(N2CCS(O)(O)CC2)ccc1-c1nc2c(N)nc(N)nc2[nH]1

nearest known ligand 0.33

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CDK1 P06493 3/20 0.32
CDK2 P24941 3/20 0.32
DHFR P00374 7/20 0.32
ADORA2A P29274 1/20 0.31
ADORA1 P30542 1/20 0.31
HRH4 Q9H3N8 2/20 0.31
TNKS O95271 1/20 0.31
PARP1 P09874 1/20 0.31
TNKS2 Q9H2K2 1/20 0.31
KDM4E B2RXH2 1/20 0.30
NPC1 O15118 1/20 0.30
RAB9A P51151 1/20 0.30
SMN1; SMN2 Q16637 1/20 0.30
CYBB P04839 1/20 0.30
NOX5 Q96PH1 1/20 0.30
NOX3 Q9HBY0 1/20 0.30
NOX4 Q9NPH5 1/20 0.30
NOX1 Q9Y5S8 1/20 0.30
ADRB1 P08588 1/20 0.30
S1PR1 P21453 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2946541 0.90 CDK1 (0.41) CDK1CDK2DHFRADORA2AADORA1
SCHEMBL2951931 0.85 PRKDC (0.42) CDK1CDK2DHFRADORA2AADORA1
SCHEMBL2953661 0.80 CDK1 (0.33) CDK1CDK2
SCHEMBL2953664 0.75
SCHEMBL3040608 0.74 F9 (0.34) ADORA2AADORA1KDM4ESMN1; SMN2
SCHEMBL2946044 0.73 MAPT (0.43) CDK1CDK2DHFRADORA2AADORA1
SCHEMBL2952943 0.72 MAP2K7 (0.45)
SCHEMBL2946546 0.71 PI4KA (0.37) CDK1CDK2DHFRHRH4
SCHEMBL2955281 0.70 CAMKK2 (0.45) ADORA2APARP1NPC1RAB9ASMN1; SMN2
SCHEMBL2946368 0.70 PRKDC (0.40) CDK1CDK2DHFRADORA2AADORA1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010111406-A2 COMPOUNDS AND THERAPEUTIC USES THEREOF MYRIAD PHARMACEUTICALS, INC. (US) 2010-09-30 WO claimed