SCHEMBL29467968

SCHEMBL29467968

NCc1ccc(N)c(F)c1F

nearest known ligand 0.39

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
LOXL2 Q9Y4K0 4/20 0.39
AOC1 P19801 2/20 0.37
AOC3 Q16853 2/20 0.37
PNMT P11086 2/20 0.34
ALDH1A1 P00352 1/20 0.32
HRH3 Q9Y5N1 1/20 0.31
MPO P05164 1/20 0.31
TAAR1 Q96RJ0 1/20 0.30
PDCD1LG2 Q9BQ51 1/20 0.30
CD274 Q9NZQ7 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13527773 0.87 LOXL2 (0.48) LOXL2AOC1AOC3PNMTHRH3
SCHEMBL5513336 0.82 ALDH1A1 (0.33) ALDH1A1
SCHEMBL961729 0.80 PNMT (0.44) LOXL2AOC1AOC3PNMTALDH1A1
SCHEMBL13743153 0.79 AOC1 (0.33) LOXL2AOC1AOC3ALDH1A1
SCHEMBL31432074 0.79 CYP3A4 (0.42) LOXL2AOC1AOC3PNMTALDH1A1
SCHEMBL27674631 0.79 LOXL2 (0.34) LOXL2AOC1AOC3PNMT
SCHEMBL20149212 0.78 FEN1 (0.37) ALDH1A1
SCHEMBL20149118 0.78 ALDH1A1 (0.31) ALDH1A1
Hydrochloric Acid SCHEMBL31431058 0.78 CYP3A4 (0.41) LOXL2AOC1AOC3PNMTALDH1A1
SCHEMBL5513611 0.78 ALDH1A1 (0.45) ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-114206870-B Tricyclic AKR1C 3-dependent KARS inhibitors 诺华股份有限公司 2024-09-03 CN disclosed
CN-114206870-A Tricyclic AKR1C3 dependent KARS inhibitors 诺华股份有限公司 2022-03-18 CN disclosed