SCHEMBL2954598

SCHEMBL2954598

COc1cc(-c2ccncc2)ccc1-c1nc2c(N)nc(N)nc2[nH]1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
DHFR P00374 3/20 0.43
DHODH Q02127 1/20 0.42
SLC2A1 P11166 1/20 0.41
AAK1 Q2M2I8 1/20 0.39
MAPK13 O15264 1/20 0.38
CYP3A4 P08684 1/20 0.38
CYP2D6 P10635 1/20 0.38
CYP2C9 P11712 1/20 0.38
SLC6A2 P23975 1/20 0.38
HTR2C P28335 1/20 0.38
ADORA2A P29274 1/20 0.38
ADORA1 P30542 1/20 0.38
MAPK12 P53778 1/20 0.38
MAPK11 Q15759 1/20 0.38
MAPK14 Q16539 1/20 0.38
TLR8 Q9NR97 1/20 0.38
TLR7 Q9NYK1 1/20 0.38
NTRK1 P04629 1/20 0.38
KIT P10721 1/20 0.37
PIK3CA P42336 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2947301 0.82 PDE2A (0.48) SLC2A1CYP3A4
SCHEMBL28861590 0.78 SLC2A1 (0.62) DHFRSLC2A1ADORA2A
SCHEMBL2952943 0.73 MAP2K7 (0.45) CYP3A4PIK3CA
SCHEMBL28861602 0.72 KDM4E (0.51) DHFRCYP2D6
SCHEMBL2946218 0.70 CHEK1 (0.47) TLR8TLR7
SCHEMBL2956342 0.69 PDE4B (0.42)
SCHEMBL27870414 0.69 PIK3CG (0.57) DHFRCYP2C9ADORA2A
SCHEMBL27870416 0.68 HEXA (0.43) DHFR
SCHEMBL2954606 0.67 HSP90AA1 (0.41) DHFR
SCHEMBL28136363 0.67 ALDH1A1 (0.74) AAK1CYP3A4TLR8TLR7NTRK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010111406-A2 COMPOUNDS AND THERAPEUTIC USES THEREOF MYRIAD PHARMACEUTICALS, INC. (US) 2010-09-30 WO claimed