SCHEMBL2947970

SCHEMBL2947970

Oc1ccc(CCN=C=S)cc1

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MIF P14174 11/20 1.00
TRPA1 O75762 2/20 0.64
CYP2E1 P05181 1/20 0.64
CYP2A6 P11509 1/20 0.64
HIF1A Q16665 1/20 0.64
CYP2A13 Q16696 1/20 0.64
EPAS1 Q99814 1/20 0.64
ESR1 P03372 1/20 0.52
ESR2 Q92731 1/20 0.52
NAAA Q02083 4/20 0.47
CA2 P00918 1/20 0.46
KDM4E B2RXH2 1/20 0.45
ALDH1A1 P00352 1/20 0.45
HTR1A P08908 1/20 0.45
ADRA2A P08913 1/20 0.45
SLC6A2 P23975 1/20 0.45
CYP2C19 P33261 1/20 0.45
HTR3A P46098 1/20 0.45
BACE1 P56817 1/20 0.45
TAAR1 Q96RJ0 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL332410 0.89 MIF (0.79) MIFTRPA1CYP2E1CYP2A6HIF1A
SCHEMBL8763660 0.83 MIF (0.70) MIFTRPA1CYP2E1CYP2A6HIF1A
SCHEMBL3364900 0.79 MIF (0.66) MIFTRPA1CYP2E1CYP2A6HIF1A
SCHEMBL3967224 0.79 MIF (0.66) MIFTRPA1CYP2E1CYP2A6HIF1A
SCHEMBL27850331 0.79 MIF (0.66) MIFTRPA1HIF1AESR1ESR2
SCHEMBL9116288 0.79 MIF (0.92) MIFTRPA1CYP2E1CYP2A6HIF1A
SCHEMBL1457483 0.79 MIF (1.00) MIFTRPA1CYP2E1CYP2A6HIF1A
SCHEMBL17971512 0.79 MIF (1.00) MIFTRPA1CYP2E1CYP2A6HIF1A
SCHEMBL30668504 0.79 MIF (1.00) MIFTRPA1CYP2E1CYP2A6HIF1A
Phenethylisothiocyanate SCHEMBL156960 0.78 MIF (1.00) MIFTRPA1CYP2E1CYP2A6HIF1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 19 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010140902-A1 INHIBITORS OF MACROPHAGE MIGRATION INHIBITORY FACTOR HAMPTON MARK (NZ) 2010-12-09 WO claimed
US-8859798-B2 Isothiocyanate compounds, pharmaceutical compositions, and uses thereof RUTGERS, THE STATE UNIVERSITY OF NEW JERSEY (US) 2014-10-14 US disclosed
US-8859798-B2 Isothiocyanate compounds, pharmaceutical compositions, and uses thereof RUTGERS, THE STATE UNIVERSITY OF NEW JERSEY (US) 2014-10-14 US disclosed
US-20090291989-A1 ISOTHIOCYANATE COMPOUNDS, PHARMACEUTICAL COMPOSITIONS, AND USES THEREOF UNIVERSITY OF MEDICINE AND DENTISTRY OF NEW JERSEY (US) 2009-11-26 US disclosed
EP-1281405-B1 Short-chained peptide-dye conjugates as contrast agents for optical diagnosis DIAGNOSTIKFORSCHUNG INST (DE) 2009-01-21 EP disclosed
US-7312326-B2 Fluorescent labeled nucleotide derivatives BECKMAN COULTER, INC. (US) 2007-12-25 US disclosed
US-7312326-B2 Fluorescent labeled nucleotide derivatives BECKMAN COULTER, INC. (US) 2007-12-25 US disclosed
US-7312326-B2 Fluorescent labeled nucleotide derivatives BECKMAN COULTER, INC. (US) 2007-12-25 US disclosed
US-7175953-B2 Short-warp peptide-dye conjugate as contrast agent for optical diagnostic INSTITUTE FUER DIAGNOSTIK FORSCHUNG (DE) 2007-02-13 US disclosed
EP-1732989-A1 FLUORESCENT LABELED NUCLEOTIDE DERIVATIVES Beckman Coulter, Inc. (US) 2006-12-20 EP disclosed
US-20060036072-A1 Short-warp peptide dye conjugate as contrast agent for optical diagnostic INSTITUT FUR DIAGNOSTIKFORSCHUNG GMBH (DE) 2006-02-16 US disclosed
WO-2005103162-A1 FLUORESCENT LABELED NUCLEOTIDE DERIVATIVES BECKMAN COULTER, INC. (US) 2005-11-03 WO disclosed
US-20050227240-A1 Fluorescent labeled nucleotide derivatives BECKMAN COULTER, INC. 2005-10-13 US disclosed
EP-1176987-B1 SHORT-CHAIN PEPTIDE DYE CONJUGATES USED AS CONTRAST AGENTS FOR OPTICAL DIAGNOSTICS DIAGNOSTIKFORSCHUNG INST (DE) 2004-02-11 EP disclosed
US-6630570-B1 Of tumor cells and tissues; derived from vaso-active intestinal protein, somatostatin or neurotensin; methine/cyanine; useful for endoscopy Insitut für Diagnostikforschung GmbH (DE) 2003-10-07 US disclosed
EP-1281405-A2 Short-chained peptide-dye conjugates as contrast agents for optical diagnosis INSTITUT FÜR DIAGNOSTIKFORSCHUNG GmbH AN DER FREIEN UNIVERSITÄT BERLIN (DE) 2003-02-05 EP disclosed
CN-1351505-A Short-chain peptide dye conjagates used as contrast agents for optical diagnostics DIAGNOSTIKFORSCHUNG INST (DE) 2002-05-29 CN disclosed
EP-1176987-A2 SHORT-CHAIN PEPTIDE DYE CONJUGATES USED AS CONTRAST AGENTS FOR OPTICAL DIAGNOSTICS INSTITUT FÜR DIAGNOSTIKFORSCHUNG GmbH AN DER FREIEN UNIVERSITÄT BERLIN (DE) 2002-02-06 EP disclosed
WO-2000061194-A2 SHORT-CHAIN PEPTIDE DYE CONJUGATES USED AS CONTRAST AGENTS FOR OPTICAL DIAGNOSTICS Institut für Diagnostikforschung GmbH an der Freien Universität Berlin (DE) 2000-10-19 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (3 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20060036072-A1 Short-warp peptide dye conjugate as contrast agent for optical diagnostic VIP, VASP, IAPP MIF 1343/4885TRPA1 1277/4885CYP2E1 4880/4885
US-20090291989-A1 ISOTHIOCYANATE COMPOUNDS, PHARMACEUTICAL COMPOSITIONS, AND USES THEREOF TST, TREH, NFATC1 MIF 545/4885TRPA1 93/4885CYP2E1 739/4885
US-20050227240-A1 Fluorescent labeled nucleotide derivatives RNGTT, DNTT, POLRMT MIF 4143/4885TRPA1 3889/4885CYP2E1 4281/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.