SCHEMBL2949173

SCHEMBL2949173

COc1ccc(-n2cnc3c(N)nc(N)nc32)c(OC)c1

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HSP90AA1 P07900 2/20 0.47
HSP90AB1 P08238 2/20 0.47
PI4KA P42356 2/20 0.45
PI4K2B Q8TCG2 2/20 0.45
PI4K2A Q9BTU6 2/20 0.45
PI4KB Q9UBF8 2/20 0.45
CDK1 P06493 2/20 0.42
CCNB1 P14635 2/20 0.42
CCNE1 P24864 2/20 0.42
CDK2 P24941 2/20 0.42
XDH P47989 2/20 0.41
MEN1 O00255 1/20 0.41
JAK2 O60674 1/20 0.41
CYP1A2 P05177 1/20 0.41
CYP3A4 P08684 1/20 0.41
GAA P10253 1/20 0.41
CYP2D6 P10635 1/20 0.41
CYP2C19 P33261 1/20 0.41
KMT2A Q03164 1/20 0.41
SMN1; SMN2 Q16637 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28861589 0.83 LMNA (0.49) HSP90AA1HSP90AB1PI4KAPI4K2BPI4K2A
SCHEMBL2954606 0.82 HSP90AA1 (0.41) HSP90AA1HSP90AB1CDK1CCNB1CCNE1
SCHEMBL28861601 0.80 PI4KA (0.68) PI4KAPI4K2BPI4K2API4KBCDK1
SCHEMBL30399128 0.80 FYN (0.41) HSP90AA1HSP90AB1GAA
SCHEMBL27870409 0.80 PI4KA (0.70) PI4KAPI4K2BPI4K2API4KBXDH
SCHEMBL2954051 0.79 DHFR (0.44) HSP90AA1HSP90AB1PI4KAPI4K2BPI4K2A
SCHEMBL2952950 0.79 DHFR (0.43) HSP90AA1HSP90AB1MEN1JAK2KMT2A
SCHEMBL2946224 0.76 CDK1 (0.40) HSP90AA1HSP90AB1CDK1CCNB1CCNE1
SCHEMBL2956345 0.75 PDE4B (0.42) HSP90AA1HSP90AB1PI4KBCDK1CDK2
SCHEMBL2953676 0.74 EGFR (0.39)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010111406-A2 COMPOUNDS AND THERAPEUTIC USES THEREOF MYRIAD PHARMACEUTICALS, INC. (US) 2010-09-30 WO claimed