SCHEMBL2956345

SCHEMBL2956345

COc1cc(C2CCN(S(C)(=O)=O)CC2)ccc1-n1cnc2c(N)nc(N)nc21

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PDE4B Q07343 1/20 0.42
EGFR P00533 6/20 0.36
CDK1 P06493 8/20 0.36
CDK4 P11802 8/20 0.36
CCND1 P24385 8/20 0.36
CDK2 P24941 8/20 0.36
HSP90AA1 P07900 1/20 0.36
HSP90AB1 P08238 1/20 0.36
CDK9 P50750 2/20 0.35
CCNT1 O60563 1/20 0.35
TP53 P04637 1/20 0.34
CASK O14936 1/20 0.34
ROCK2 O75116 1/20 0.34
CDKL5 O76039 1/20 0.34
STK10 O94804 1/20 0.34
CDK14 O94921 1/20 0.34
ABL1 P00519 1/20 0.34
MAK P20794 1/20 0.34
CDK11B P21127 1/20 0.34
TTK P33981 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2946285 0.90 PDE4B (0.46) PDE4BHSP90AA1HSP90AB1CDK9CCNT1
SCHEMBL2946224 0.85 CDK1 (0.40) CDK1CDK2HSP90AA1HSP90AB1CAMK2D
SCHEMBL2948407 0.83 PIK3CD (0.40) TTK
SCHEMBL2946341 0.81 PIK3CD (0.39) EGFRTTK
SCHEMBL2950527 0.79 ADORA2A (0.42) CDK1CDK2HSP90AA1HSP90AB1
SCHEMBL2949173 0.75 HSP90AA1 (0.47) CDK1CDK2HSP90AA1HSP90AB1PI4KB
SCHEMBL2956342 0.74 PDE4B (0.42) PDE4BEGFRCDK1CDK4CCND1
SCHEMBL2953676 0.74 EGFR (0.39) EGFRCDK4CCND1CDK9CCNT1
SCHEMBL17197373 0.73 PDE4B (0.57) PDE4BEGFRCDK9CCNT1TP53
SCHEMBL2953257 0.72 CDK1 (0.42) CDK1CDK2PI4KB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010111406-A2 COMPOUNDS AND THERAPEUTIC USES THEREOF MYRIAD PHARMACEUTICALS, INC. (US) 2010-09-30 WO claimed