SCHEMBL2952950

SCHEMBL2952950

COc1cc(N2CCOCC2)ccc1-n1cnc2c(N)nc(N)nc21

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
DHFR P00374 3/20 0.43
INSR P06213 1/20 0.41
ALK Q9UM73 1/20 0.41
FYN P06241 1/20 0.41
LRRK2 Q5S007 1/20 0.40
PIK3CA P42336 2/20 0.40
SIK1 P57059 1/20 0.40
SIK2 Q9H0K1 1/20 0.40
SIK3 Q9Y2K2 1/20 0.40
MEN1 O00255 1/20 0.39
THRB P10828 1/20 0.39
KMT2A Q03164 1/20 0.39
MTOR P42345 1/20 0.39
TTK P33981 3/20 0.39
SUV39H2 Q9H5I1 1/20 0.39
JAK2 O60674 1/20 0.39
HSP90AA1 P07900 1/20 0.39
HSP90AB1 P08238 1/20 0.39
KIT P10721 1/20 0.39
FLT3 P36888 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2946049 0.91 DHFR (0.42) DHFRTTK
SCHEMBL2953119 0.91 TTK (0.43) INSRALKTTKFLT3
SCHEMBL2954051 0.90 DHFR (0.44) DHFRHSP90AA1HSP90AB1
SCHEMBL30399128 0.89 FYN (0.41) DHFRFYNHSP90AA1HSP90AB1FLT3
SCHEMBL2952940 0.87 SMPD3 (0.41) INSRALKTTK
SCHEMBL2951937 0.86 DHFR (0.45) DHFRPIK3CAMEN1KMT2AMTOR
SCHEMBL2953492 0.84 TTK (0.47) ALKPIK3CAMTORTTK
SCHEMBL2948890 0.83 TTK (0.45) DHFRINSRALKPIK3CATTK
SCHEMBL2953676 0.82 EGFR (0.39) DHFRALKFYNFLT3
SCHEMBL2946373 0.82 DHFR (0.43) DHFRPIK3CAMTOR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010111406-A2 COMPOUNDS AND THERAPEUTIC USES THEREOF MYRIAD PHARMACEUTICALS, INC. (US) 2010-09-30 WO claimed
CN-116284001-A DCLK1 inhibitor, preparation method, pharmaceutical composition and application 中国药科大学 2023-06-23 CN disclosed