SCHEMBL29519663

SCHEMBL29519663

N#Cc1ccc(-c2cccc(F)c2)c(C2CC2)c1

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GABRG2 P18507 2/20 0.43
GABRB3 P28472 2/20 0.43
GABRA5 P31644 2/20 0.43
GABRA3 P34903 2/20 0.43
CHRNA1 P02708 1/20 0.41
CHRNG P07510 1/20 0.41
CHRNB1 P11230 1/20 0.41
CHRNB2 P17787 1/20 0.41
CHRNB4 P30926 1/20 0.41
CHRNA3 P32297 1/20 0.41
CHRNA4 P43681 1/20 0.41
CHRND Q07001 1/20 0.41
KDM4E B2RXH2 1/20 0.41
HPGD P15428 1/20 0.41
NPSR1 Q6W5P4 1/20 0.41
RXFP1 Q9HBX9 1/20 0.41
CYP11B2 P19099 5/20 0.40
CYP11B1 P15538 2/20 0.40
KDM1A O60341 1/20 0.40
CHEK1 O14757 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4965411 0.79 PTGDR2 (0.45) CHRNA1CHRNGCHRNB1CHRNB2CHRNB4
SCHEMBL27626880 0.78 PTGDR2 (0.50) CHRNA1CHRNGCHRNB1CHRNB2CHRNB4
SCHEMBL25259090 0.77 KDM1A (0.39) CHRNA1CHRNGCHRNB1CHRNB2CHRNB4
SCHEMBL30591409 0.77 KDM1A (0.39) CHRNA1CHRNGCHRNB1CHRNB2CHRNB4
SCHEMBL29430712 0.77 GABRG2 (0.46) GABRG2GABRB3GABRA5GABRA3KDM4E
SCHEMBL5098919 0.75 MAOA (0.48) GABRG2GABRB3GABRA5GABRA3KDM4E
SCHEMBL16905570 0.75 CHRNA1 (0.65) CHRNA1CHRNGCHRNB1CHRNB2CHRNB4
SCHEMBL22637087 0.75 ACLY (0.42) GRM5
SCHEMBL2695090 0.74 CHRNA1 (0.46) CHRNA1CHRNGCHRNB1CHRNB2CHRNB4
SCHEMBL10865411 0.72 CYP11B2 (0.36) CHRNA1CHRNGCHRNB1CHRNB2CHRNB4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-109743875-B Inhibitors of the MENIN-MLL interaction 生命医药有限责任公司 2022-04-29 CN disclosed