SCHEMBL4965411

SCHEMBL4965411

N#Cc1ccc(-c2ccccc2)c(C2CCC2)c1

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PTGDR2 Q9Y5Y4 2/20 0.45
CYP11B2 P19099 2/20 0.44
NOS3 P29474 1/20 0.40
NOS1 P29475 1/20 0.40
NOS2 P35228 1/20 0.40
DRD2 P14416 3/20 0.40
DRD3 P35462 3/20 0.40
KDM4E B2RXH2 1/20 0.40
MEN1 O00255 1/20 0.40
ALDH1A1 P00352 1/20 0.40
MAPT P10636 1/20 0.40
HPGD P15428 1/20 0.40
TSHR P16473 1/20 0.40
KMT2A Q03164 1/20 0.40
NPSR1 Q6W5P4 1/20 0.40
HSD17B10 Q99714 1/20 0.40
CHRNA1 P02708 1/20 0.40
CHRNG P07510 1/20 0.40
CHRNB1 P11230 1/20 0.40
CHRNB2 P17787 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27626880 0.95 PTGDR2 (0.50) PTGDR2CYP11B2NOS3NOS1NOS2
SCHEMBL10865411 0.80 CYP11B2 (0.36) PTGDR2CYP11B2DRD2DRD3KDM4E
SCHEMBL29519663 0.79 GABRG2 (0.43) CYP11B2KDM4EHPGDNPSR1CHRNA1
SCHEMBL27450587 0.78 CYP11B2 (0.35) PTGDR2CYP11B2DRD2DRD3KDM4E
SCHEMBL28442339 0.78 CNR1 (0.39) PTGDR2CYP11B2KDM4EMEN1ALDH1A1
SCHEMBL15767956 0.77 GRIA1 (0.37) PTGDR2CYP11B2DRD2DRD3KDM4E
SCHEMBL16905238 0.76 CHRNA1 (0.59) PTGDR2CYP11B2NOS3NOS1NOS2
SCHEMBL27626879 0.76 PTGS2 (0.56) PTGDR2CYP11B2ALDH1A1CYP19A1CYP11B1
SCHEMBL10606461 0.76 KDM1A (0.45) PTGDR2CYP11B2DRD2DRD3TSHR
SCHEMBL4983356 0.75 CHRNB2 (0.40) PTGDR2CYP11B2MEN1ALDH1A1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1888523-A2 CYCLOBUTYL AMINE DERIVATIVES Abbott Laboratories (US) 2008-02-20 EP disclosed
WO-2006132914-A2 CYCLOBUTYL AMINE DERIVATIVES ABBOTT LABORATORIES (US) 2006-12-14 WO disclosed