SCHEMBL2948890

SCHEMBL2948890

COc1cc(N2CCN(CC3CCOC3)CC2)ccc1-n1cnc2c(N)nc(N)nc21

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TTK P33981 2/20 0.45
TLR7 Q9NYK1 2/20 0.40
TLR9 Q9NR96 1/20 0.40
TLR8 Q9NR97 1/20 0.40
PIK3CA P42336 2/20 0.37
ENPP2 Q13822 3/20 0.35
HTR1A P08908 4/20 0.35
HTR7 P34969 3/20 0.34
HSP90AA1 P07900 1/20 0.34
HSP90AB1 P08238 1/20 0.34
DHFR P00374 1/20 0.34
ADRA1D P25100 2/20 0.34
ADRA1A P35348 2/20 0.34
ADRA1B P35368 2/20 0.34
PDE10A Q9Y233 2/20 0.34
PDE1B Q01064 1/20 0.34
BRAF P15056 1/20 0.33
ACVR1 Q04771 1/20 0.33
INSR P06213 1/20 0.33
IGF1R P08069 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2952950 0.83 DHFR (0.43) TTKPIK3CAHSP90AA1HSP90AB1DHFR
SCHEMBL2953119 0.81 TTK (0.43) TTKACVR1INSRIGF1RALK
SCHEMBL30399128 0.81 FYN (0.41) HSP90AA1HSP90AB1DHFR
SCHEMBL2954051 0.80 DHFR (0.44) HSP90AA1HSP90AB1DHFR
SCHEMBL2950126 0.78 TTK (0.42) TTKHTR7HSP90AA1HSP90AB1DHFR
SCHEMBL2952940 0.78 SMPD3 (0.41) TTKINSRIGF1RALK
SCHEMBL3034636 0.77 HSP90AA1 (0.38) HSP90AA1HSP90AB1INSRIGF1RALK
SCHEMBL2946049 0.77 DHFR (0.42) TTKDHFR
SCHEMBL2953492 0.76 TTK (0.47) TTKPIK3CAALK
SCHEMBL2953676 0.75 EGFR (0.39) DHFRALK

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010111406-A2 COMPOUNDS AND THERAPEUTIC USES THEREOF MYRIAD PHARMACEUTICALS, INC. (US) 2010-09-30 WO claimed