SCHEMBL29558689

SCHEMBL29558689

COc1ccc(Cc2nc(N)ncc2N)cc1

nearest known ligand 0.64

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.54
CYP2D6 P10635 1/20 0.54
ATM Q13315 1/20 0.54
POLB P06746 1/20 0.54
DHFR P00374 2/20 0.48
KMT2A Q03164 1/20 0.48
CSF1R P07333 2/20 0.47
NTRK2 Q16620 2/20 0.47
NTRK1 P04629 1/20 0.47
NTRK3 Q16288 1/20 0.47
NPSR1 Q6W5P4 1/20 0.47
CDC25A P30304 1/20 0.46
CDC25B P30305 1/20 0.46
PDE3B Q13370 1/20 0.46
PDE3A Q14432 1/20 0.46
PDE10A Q9Y233 1/20 0.46
PKM P14618 1/20 0.46
LMNA P02545 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10698612 0.78 MPO (0.47) CYP2D6
SCHEMBL11567058 0.78 ALDH1A1 (0.57) ALDH1A1CYP2D6ATMPOLBDHFR
SCHEMBL28362594 0.78 DHFR (0.55) ALDH1A1CYP2D6ATMPOLBDHFR
SCHEMBL8376680 0.78 DHFR (0.76) DHFRCSF1RNTRK2NTRK1NTRK3
SCHEMBL28585742 0.76 ALDH1A1 (0.64) ALDH1A1CYP2D6ATMPOLBKMT2A
SCHEMBL28528829 0.76 ALDH1A1 (0.69) ALDH1A1CYP2D6ATMPOLBDHFR
SCHEMBL23612255 0.75 ALDH1A1 (0.82) ALDH1A1CYP2D6ATMDHFRNPSR1
SCHEMBL30055740 0.75 ALDH1A1 (0.82) ALDH1A1CYP2D6ATMDHFRNPSR1
SCHEMBL28802706 0.75 ALDH1A1 (0.54) ALDH1A1CYP2D6ATMPOLBNPSR1
SCHEMBL23392698 0.75 APP (0.59) POLBKMT2ALMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-111943892-B Histone deacetylase subtype inhibitor thioacetylarylamine compound and application thereof 上海中泽医药科技有限公司 2022-04-05 CN disclosed