SCHEMBL2946285

SCHEMBL2946285

COc1cc(C2CCCN(S(C)(=O)=O)C2)ccc1-n1cnc2c(N)nc(N)nc21

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PDE4B Q07343 4/20 0.46
ALDH1A1 P00352 1/20 0.40
LMNA P02545 1/20 0.40
PIK3CD O00329 1/20 0.37
PIK3R1 P27986 1/20 0.37
PIK3CA P42336 1/20 0.37
PIK3CB P42338 1/20 0.37
ADORA2A P29274 1/20 0.36
KMT2A Q03164 2/20 0.34
HSP90AA1 P07900 1/20 0.34
HSP90AB1 P08238 1/20 0.34
POLB P06746 1/20 0.33
SMN1; SMN2 Q16637 1/20 0.33
RAB9A P51151 1/20 0.33
CCNT1 O60563 1/20 0.33
CDK9 P50750 1/20 0.33
DRD2 P14416 1/20 0.33
DRD1 P21728 1/20 0.33
DRD4 P21917 1/20 0.33
DRD5 P21918 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2956345 0.90 PDE4B (0.42) PDE4BHSP90AA1HSP90AB1CCNT1CDK9
SCHEMBL2950527 0.85 ADORA2A (0.42) ADORA2AHSP90AA1HSP90AB1DRD2DRD1
SCHEMBL2946224 0.79 CDK1 (0.40) HSP90AA1HSP90AB1DRD3
SCHEMBL2946279 0.76 PDE4B (0.46) PDE4BALDH1A1LMNAPIK3CDPIK3R1
SCHEMBL2948407 0.75 PIK3CD (0.40) ALDH1A1LMNAPIK3CDPIK3R1PIK3CA
SCHEMBL2946341 0.75 PIK3CD (0.39) ALDH1A1PIK3CDPIK3R1PIK3CAPIK3CB
SCHEMBL2949173 0.72 HSP90AA1 (0.47) KMT2AHSP90AA1HSP90AB1SMN1; SMN2
SCHEMBL2950550 0.71 CYP1A2 (0.50) PIK3R1PIK3CAADORA2ASMN1; SMN2
SCHEMBL2953676 0.71 EGFR (0.39) CCNT1CDK9
SCHEMBL2952077 0.71 INSR (0.42) KMT2AHSP90AA1HSP90AB1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010111406-A2 COMPOUNDS AND THERAPEUTIC USES THEREOF MYRIAD PHARMACEUTICALS, INC. (US) 2010-09-30 WO claimed