SCHEMBL2957014

SCHEMBL2957014

CC(=O)Nc1ccc(S(=O)(=O)N2CCN(c3ccccc3)CC2)cc1

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
MAPT P10636 3/20 1.00
KMT2A Q03164 7/20 0.82
MEN1 O00255 5/20 0.82
F13A1 P00488 1/20 0.72
TGM2 P21980 1/20 0.72
TGM1 P22735 1/20 0.72
ATM Q13315 1/20 0.69
L3MBTL1 Q9Y468 1/20 0.67
ALDH1A1 P00352 2/20 0.66
HPGD P15428 1/20 0.66
GAA P10253 2/20 0.65
HTT P42858 1/20 0.65
SMN1; SMN2 Q16637 1/20 0.65
USP2 O75604 1/20 0.64
LMNA P02545 1/20 0.64
PKM P14618 1/20 0.64

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1662361 0.86 MAPT (0.74) MAPTKMT2AMEN1F13A1TGM2
SCHEMBL1874408 0.84 F13A1 (1.00) MAPTF13A1TGM2TGM1ALDH1A1
SCHEMBL23217100 0.83 MAPT (0.70) MAPTKMT2AMEN1ATMALDH1A1
SCHEMBL4759272 0.82 KMT2A (0.78) MAPTKMT2AMEN1L3MBTL1ALDH1A1
SCHEMBL3300404 0.82 ALDH1A1 (0.84) MAPTKMT2AMEN1L3MBTL1ALDH1A1
SCHEMBL30513335 0.81 SMN1; SMN2 (0.79) MAPTKMT2AMEN1ALDH1A1GAA
SCHEMBL18711452 0.81 KMT2A (0.76) MAPTKMT2AMEN1L3MBTL1ALDH1A1
SCHEMBL4075002 0.81 L3MBTL1 (1.00) MAPTKMT2AMEN1L3MBTL1ALDH1A1
SCHEMBL4070839 0.80 ALDH1A1 (0.84) MAPTKMT2AMEN1L3MBTL1ALDH1A1
SCHEMBL616835 0.80 ALDH1A1 (0.78) MAPTKMT2AMEN1L3MBTL1ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 11 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7759339-B2 Hydroxysteroid dehydrogenase inhibitors TAKEDA SAN DIEGO, INC. (US) 2010-07-20 US claimed
EP-1866298-A2 HYDROXYSTEROID DEHYDROGENASE INHIBITORS Takeda San Diego, Inc. (US) 2007-12-19 EP claimed
WO-2006105127-A2 HYDROXYSTEROID DEHYDROGENASE INHIBITORS TAKEDA SAN DIEGO, INC. (US) 2006-10-05 WO claimed
US-20060223829-A1 Hydroxysteroid dehydrogenase inhibitors TAKEDA SAN DIEGO, INC. 2006-10-05 US claimed
CN-119330892-A Benzenesulfonamide derivative and preparation method and application thereof 天津科技大学 2025-01-21 CN disclosed
CN-116496292-A Benzenesulfonamide derivative and preparation method and application thereof 天津科技大学 2023-07-28 CN disclosed
US-7759339-B2 Hydroxysteroid dehydrogenase inhibitors TAKEDA SAN DIEGO, INC. (US) 2010-07-20 US disclosed
US-7759339-B2 Hydroxysteroid dehydrogenase inhibitors TAKEDA SAN DIEGO, INC. (US) 2010-07-20 US disclosed
EP-1866298-A2 HYDROXYSTEROID DEHYDROGENASE INHIBITORS Takeda San Diego, Inc. (US) 2007-12-19 EP disclosed
WO-2006105127-A2 HYDROXYSTEROID DEHYDROGENASE INHIBITORS TAKEDA SAN DIEGO, INC. (US) 2006-10-05 WO disclosed
US-20060223829-A1 Hydroxysteroid dehydrogenase inhibitors TAKEDA SAN DIEGO, INC. 2006-10-05 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20060223829-A1 Hydroxysteroid dehydrogenase inhibitors HSD17B1, HSD17B3, HSD17B2 MAPT 3168/4885KMT2A 3335/4885MEN1 2689/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.