Argatroban

Argatroban

SCHEMBL29618936

CC1CNc2c(cccc2S(=O)(=O)N[C@@H](CCCN=C(N)N)C(=O)N2CC[C@@H](C)C[C@@H]2C(=O)O)C1.O

nearest known ligand 0.99

Full drug profile on Sugi Atlas →

Known targets — ChEMBL curated mechanism

F2

The experimentally established mechanism targets of Argatroban. The predicted profile below is derived independently by chemical similarity — agreement is a validation signal, a miss is honest.

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
F2 known ✓ P00734 4/20 0.99
PRSS1 P07477 2/20 0.99
F10 P00742 2/20 0.99
LMNA P02545 1/20 0.99
PLAT P00750 1/20 0.99
PRSS2 P07478 1/20 0.99
PRSS3 P35030 1/20 0.99

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Argatroban SCHEMBL20787652 1.00 F2 (0.99) F2PRSS1F10LMNAPLAT
Argatroban SCHEMBL135173 0.99 F2 (1.00) F2PRSS1F10LMNAPLAT
Argatroban SCHEMBL22974994 0.99 F2 (1.00) F2PRSS1F10LMNAPLAT
Argatroban SCHEMBL18895186 0.99 F2 (1.00) F2PRSS1F10LMNAPLAT
Argatroban SCHEMBL4375 0.99 F2 (1.00) F2PRSS1F10LMNAPLAT
Argatroban SCHEMBL29741503 0.99 F2 (1.00) F2PRSS1F10LMNAPLAT
Argatroban SCHEMBL20567702 0.99 F2 (1.00) F2PRSS1F10LMNAPLAT
Argatroban SCHEMBL15019460 0.99 F2 (1.00) F2PRSS1F10LMNAPLAT
SCHEMBL24209448 0.94 F2 (0.90) F2PRSS1F10LMNAPLAT
SCHEMBL29566356 0.90 F2 (0.84) F2PRSS1F10LMNAPLAT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 25 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20260131014-A1 SUPRAMOLECULAR AGENTS DESIGN & USES THEREOF UNIV GENEVE (CH) 2026-05-14 US disclosed
EP-4658228-A1 ECO-BIOLOGICAL COSMETIC COMPOSITION SUITABLE FOR REDUCING THE SIGNS OF CUTANEOUS AGEING Thorel, Jean-Noël (FR) 2025-12-10 EP disclosed
EP-3927817-B1 NEW RECOMBINANT DIAMINE OXIDASE AND ITS USE FOR THE TREATMENT OF DISEASES CHARACTERIZED BY EXCESS HISTAMINE UNIV WIEN MED (AT) 2025-08-20 EP disclosed
US-20250073210-A1 Use of Ergothioneine for Enhancing Glutathione Level NANJING NUTRABUILDING BIO TECH CO LTD (CN) 2025-03-06 US disclosed
EP-4460300-A1 USE OF ERGOTHIONEINE FOR ENHANCING GLUTATHIONE LEVEL Nanjing Nutrabuilding Bio-Tech Co., Ltd. (CN) 2024-11-13 EP disclosed
US-20240366496-A1 COSMETIC COMPOSITION COMPRISING AT LEAST ONE BIRCH EXTRACT AND AT LEAST ONE BEECH BUD EXTRACT CREDO (FR) 2024-11-07 US disclosed
WO-2024186730-A1 COMPOSITIONS FOR ENHANCED METABOLIC OXIDATION OF FATTY ACIDS GRADS INNOVATION (US) 2024-09-12 WO disclosed
CN-118510508-A Use of ergothioneine for increasing glutathione levels 南京纽邦生物科技有限公司 2024-08-16 CN disclosed
WO-2024161085-A1 ECO-BIOLOGICAL COSMETIC COMPOSITION SUITABLE FOR REDUCING THE SIGNS OF CUTANEOUS AGEING NAOS INSTITUTE OF LIFE SCIENCE (FR) 2024-08-08 WO disclosed
US-20240215579-A1 USE OF ANTI-CLOTTING COMPOUNDS AS RODENTICIDES GULBA DIETRICH (DE) 2024-07-04 US disclosed
US-20230226070-A1 TREATMENT OF THROMBOSIS AND ASSOCIATED DISORDERS WITH AN ANTI-PLATELET AGENT. THE HEART RESEARCH INSTITUTE LTD (AU) 2023-07-20 US disclosed
WO-2023131078-A1 USE OF ERGOTHIONEINE FOR ENHANCING GLUTATHIONE LEVEL NANJING NUTRABUILDING BIO-TECH CO., LTD. (CN) 2023-07-13 WO disclosed
US-11678659-B2 Use as rodenticides of compounds that inhibit blood coagulation GULBA DIETRICH (DE) 2023-06-20 US disclosed
WO-2023089288-A1 COSMETIC AND/OR DERMATOLOGICAL COMPOSITION COMPRISING AT LEAST ONE EXTRACT OF CYLINDROTHECA FUSIFORMIS AND AT LEAST ONE EXTRACT OF DUNALIELLA SALINA, AND COSMETIC USES THEREOF BLUE LAB (FR) 2023-05-25 WO disclosed
EP-4149477-A1 TREATMENT OF THROMBOSIS AND ASSOCIATED DISORDERS WITH AN ANTI-PLATELET AGENT The Heart Research Institute Ltd (AU) 2023-03-22 EP disclosed
US-11491141-B1 Methods of treating glutathione deficiencies and deficiencies in glutathione synthetase activity NANJING NUTRABUILDING BIO-TECH CO., LTD. (CN) 2022-11-08 US disclosed
WO-2022214485-A1 USE OF ANTI-CLOTTING COMPOUNDS AS RODENTICIDES BIOROXX GMBH (DE) 2022-10-13 WO disclosed
EP-4070658-A1 USE OF ANTICOAGULANT ACTIVE COMPOUNDS AS RODENTICIDE BIORoxx GmbH (DE) 2022-10-12 EP disclosed
WO-2022208005-A1 COSMETIC COMPOSITION COMPRISING AT LEAST ONE BIRCH EXTRACT AND AT LEAST ONE BEECH BUD EXTRACT CREDO (FR) 2022-10-06 WO disclosed
US-20220145269-A1 NEW RECOMBINANT DIAMINE OXIDASE AND ITS USE FOR THE TREATMENT OF DISEASES CHARACTERIZED BY EXCESS HISTAMINE UNIVERSITÄT FÜR BODENKULTUR WIEN (AT) 2022-05-12 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (6 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-11491141-B1 Methods of treating glutathione deficiencies and deficiencies in glutathione synthetase activity GSS, GGT1, GSTA2 F2 3396/4885PRSS1 323/4885F10 4389/4885
US-11678659-B2 Use as rodenticides of compounds that inhibit blood coagulation PLAT, F2R, PLAUR F2 11/4885PRSS1 199/4885F10 53/4885
US-20230226070-A1 TREATMENT OF THROMBOSIS AND ASSOCIATED DISORDERS WITH AN ANTI-PLATELET AGENT. PLAT, PLA2G7, PIK3R5 F2 219/4885PRSS1 139/4885F10 286/4885
US-20250073210-A1 Use of Ergothioneine for Enhancing Glutathione Level GSS, GPX1, GSTA1 F2 3386/4885PRSS1 349/4885F10 4334/4885
US-20240215579-A1 USE OF ANTI-CLOTTING COMPOUNDS AS RODENTICIDES PLG, F13B, F2 F2 3/4885PRSS1 175/4885F10 30/4885
US-20260131014-A1 SUPRAMOLECULAR AGENTS DESIGN & USES THEREOF ADAR, RBM39, ANTXR2 F2 94/4885PRSS1 3359/4885F10 837/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.