SCHEMBL2962655

SCHEMBL2962655

CC1=Cc2c(cc(Br)cc2-c2ccccc2)C1

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
AKR1C3 P42330 1/20 0.38
AKR1C2 P52895 1/20 0.38
AKR1C1 Q04828 1/20 0.38
ESR2 Q92731 1/20 0.36
ALDH1A1 P00352 3/20 0.34
MAPK1 P28482 2/20 0.34
PDE4B Q07343 1/20 0.32
NPC1 O15118 1/20 0.32
TSHR P16473 1/20 0.32
RAB9A P51151 1/20 0.32
PTGDR2 Q9Y5Y4 1/20 0.32
ALOX5 P09917 1/20 0.32
GABRA1 P14867 2/20 0.32
GABRA5 P31644 2/20 0.32
GABRA2 P47869 2/20 0.32
GABRB2 P47870 2/20 0.32
MAOB P27338 3/20 0.31
BACE1 P56817 1/20 0.31
GABRG2 P18507 1/20 0.31
GABRB3 P28472 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2965828 0.89 ESR1 (0.34) ESR2ALDH1A1NPC1RAB9AKDM4E
SCHEMBL4203318 0.83 PSMB5 (0.38) ESR2ALDH1A1MAPK1TSHRPTGDR2
SCHEMBL2482030 0.80 DHODH (0.37) ESR2PTGDR2CYP2A6NPSR1
SCHEMBL2963372 0.79 AKR1C3 (0.33) AKR1C3AKR1C2AKR1C1PDE4BPTGDR2
SCHEMBL2962116 0.79 HSD11B1 (0.38) ALDH1A1MAPK1NPC1RAB9APSMB5
SCHEMBL4653379 0.78 METAP2 (0.41) AKR1C3AKR1C2AKR1C1ESR2TSHR
SCHEMBL29949127 0.78 ALDH1A1 (0.33) ESR2ALDH1A1NPC1RAB9A
SCHEMBL14645967 0.78 ALDH1A1 (0.33) ESR2ALDH1A1NPC1RAB9A
SCHEMBL2969288 0.77 KDM4E (0.35) ALDH1A1MAOBCYP2A6KDM4E
SCHEMBL2963190 0.76 KDM4E (0.31) MAOBKDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 8 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7767818-B2 Hepatitis C inhibitor dipeptide analogs BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2010-08-03 US disclosed
US-7763562-B2 Heteroatom bridged metallocene compounds for olefin polymerization EXXONMOBIL CHEMICAL PATENTS INC. (US) 2010-07-27 US disclosed
US-7696242-B2 Hepatitis C inhibitor peptide analogs BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2010-04-13 US disclosed
US-20090156822-A1 Hepatitis C Inhibitor Dipeptide Analogs BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2009-06-18 US disclosed
US-7511157-B2 racemic mixtures, stereoisomers or optical isomers, useful as protease inhibitors; viricides BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2009-03-31 US disclosed
US-20070135597-A1 Heteroatom bridged metallocene compounds for olefin polymerization EXXONMOBIL CHEMICAL PATENTS INC. 2007-06-14 US disclosed
WO-2006065809-A2 HETEROATOM BRIDGED METALLOCENE COMPOUNDS FOR OLEFIN POLYMERIZATION EXXONMOBIL CHEMICAL PATENTS INC. (US) 2006-06-22 WO disclosed
US-20060019905-A1 inhibitors of the hepatitis C virus NS3 protease; azalactone intermediate reacted with cycloalkylsulfonamide and decylization; urea or carbamate-terminated alkylglycine, hydroxyproline, cyclopropylglycine tripeptide BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2006-01-26 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (3 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20090156822-A1 Hepatitis C Inhibitor Dipeptide Analogs DPP3, CTSC, ANPEP AKR1C3 773/4885AKR1C2 1891/4885AKR1C1 1582/4885
US-20070135597-A1 Heteroatom bridged metallocene compounds for olefin polymerization AP2M1, AP1M1, PYM1 AKR1C3 3611/4885AKR1C2 3868/4885AKR1C1 4022/4885
US-20060019905-A1 inhibitors of the hepatitis C virus NS3 protease; azalactone intermediate reacted with cycloalkylsulfonamide and decylization; urea or carbamate-terminated alkylglycine, hydroxyproline, cyclopropylglycine tripeptide CPN1, HPN, CTSC AKR1C3 1276/4885AKR1C2 1760/4885AKR1C1 1525/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.