SCHEMBL2962903

SCHEMBL2962903

NC(=O)c1ccccc1N1CCN(S(=O)(=O)c2ccccc2Cl)CC1

nearest known ligand 0.55

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 1/20 0.55
CHRM4 P08173 3/20 0.51
HSD11B1 P28845 1/20 0.48
KMT2A Q03164 2/20 0.46
FAAH O00519 2/20 0.46
ALDH1A1 P00352 4/20 0.45
LMNA P02545 3/20 0.45
SMN1; SMN2 Q16637 3/20 0.45
RPS6KB1 P23443 1/20 0.45
GBA1 P04062 1/20 0.45
TP53 P04637 1/20 0.45
TSHR P16473 1/20 0.45
HSD17B10 Q99714 1/20 0.45
MAPT P10636 2/20 0.44
HTT P42858 2/20 0.44
GAA P10253 1/20 0.44
PKM P14618 1/20 0.44
MAPK1 P28482 1/20 0.44
HDAC3 O15379 1/20 0.44
HDAC4 P56524 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2959432 0.88 CHRM4 (0.52) CHRM4HSD11B1KMT2AFAAHALDH1A1
SCHEMBL2961026 0.84 CHRM4 (0.62) CHRM4HSD11B1KMT2AALDH1A1LMNA
SCHEMBL2961967 0.81 ALDH1A1 (0.61) CHRM4HSD11B1KMT2AFAAHALDH1A1
SCHEMBL2963243 0.81 CHRM4 (0.56) CHRM4HSD11B1KMT2AALDH1A1LMNA
SCHEMBL3223609 0.79 CHRM4 (0.57) CHRM4HSD11B1KMT2ALMNAGBA1
SCHEMBL5331434 0.79 CHRM4 (0.64) CHRM4HSD11B1KMT2AALDH1A1LMNA
SCHEMBL3216764 0.78 ALDH1A1 (0.64) CHRM4HSD11B1KMT2AALDH1A1LMNA
SCHEMBL10723724 0.78 CHRM4 (0.64) CHRM4KMT2AFAAHALDH1A1LMNA
SCHEMBL2953059 0.75 CHRM4 (0.53) CHRM4HSD11B1ALDH1A1GBA1GAA
SCHEMBL2950399 0.75 SMN1; SMN2 (0.74) KMT2AALDH1A1LMNASMN1; SMN2TP53

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 10 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7759339-B2 Hydroxysteroid dehydrogenase inhibitors TAKEDA SAN DIEGO, INC. (US) 2010-07-20 US claimed
EP-1866298-A2 HYDROXYSTEROID DEHYDROGENASE INHIBITORS Takeda San Diego, Inc. (US) 2007-12-19 EP claimed
WO-2006105127-A2 HYDROXYSTEROID DEHYDROGENASE INHIBITORS TAKEDA SAN DIEGO, INC. (US) 2006-10-05 WO claimed
US-20060223829-A1 Hydroxysteroid dehydrogenase inhibitors TAKEDA SAN DIEGO, INC. 2006-10-05 US claimed
US-7759339-B2 Hydroxysteroid dehydrogenase inhibitors TAKEDA SAN DIEGO, INC. (US) 2010-07-20 US disclosed
US-7759339-B2 Hydroxysteroid dehydrogenase inhibitors TAKEDA SAN DIEGO, INC. (US) 2010-07-20 US disclosed
US-7759339-B2 Hydroxysteroid dehydrogenase inhibitors TAKEDA SAN DIEGO, INC. (US) 2010-07-20 US disclosed
EP-1866298-A2 HYDROXYSTEROID DEHYDROGENASE INHIBITORS Takeda San Diego, Inc. (US) 2007-12-19 EP disclosed
WO-2006105127-A2 HYDROXYSTEROID DEHYDROGENASE INHIBITORS TAKEDA SAN DIEGO, INC. (US) 2006-10-05 WO disclosed
US-20060223829-A1 Hydroxysteroid dehydrogenase inhibitors TAKEDA SAN DIEGO, INC. 2006-10-05 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20060223829-A1 Hydroxysteroid dehydrogenase inhibitors HSD17B1, HSD17B3, HSD17B2 NPC1 762/4885CHRM4 4346/4885HSD11B1 7/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.