SCHEMBL29630932

SCHEMBL29630932

Cc1cccc(-n2ccc3c(=O)[nH]cnc32)n1

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TGFBR1 P36897 5/20 0.47
GAA P10253 1/20 0.42
PARP1 P09874 7/20 0.42
RECQL P46063 1/20 0.40
ALDH1A1 P00352 1/20 0.39
ALOX5 P09917 1/20 0.37
HTT P42858 1/20 0.36
PDPK1 O15530 1/20 0.36
CA12 O43570 1/20 0.36
ALOX15 P16050 1/20 0.36
SMN1; SMN2 Q16637 1/20 0.36
CA9 Q16790 1/20 0.36
TNKS2 Q9H2K2 1/20 0.36
LMNA P02545 1/20 0.36
MAPT P10636 1/20 0.36
KMT2A Q03164 1/20 0.36
AURKA O14965 1/20 0.36
DAPK3 O43293 1/20 0.36
JAK2 O60674 1/20 0.36
PRKD3 O94806 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20971165 1.00 TGFBR1 (0.47) TGFBR1GAAPARP1RECQLALDH1A1
SCHEMBL29630995 0.83 ALOX5 (0.41) TGFBR1PARP1ALDH1A1ALOX5PDPK1
SCHEMBL20971154 0.83 ALOX5 (0.41) TGFBR1PARP1ALDH1A1ALOX5PDPK1
SCHEMBL19692167 0.79 GAA (0.47) GAAPARP1ALDH1A1HTTPDPK1
SCHEMBL29627428 0.79 GAA (0.47) GAAPARP1ALDH1A1HTTPDPK1
SCHEMBL20971046 0.76 LMNA (0.58) PARP1ALDH1A1HTTLMNAMAPT
SCHEMBL20971226 0.75 PARP1 (0.48) PARP1ALDH1A1HTTPDPK1CA12
SCHEMBL29631014 0.75 PARP1 (0.48) PARP1ALDH1A1HTTPDPK1CA12
SCHEMBL20971305 0.74 MAPT (0.53) PARP1ALDH1A1HTTLMNAMAPT
SCHEMBL19692323 0.74 ALDH1A1 (0.43) PARP1ALDH1A1HTTPDPK1CA12

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-109563094-B (hetero) aryl-substituted piperidinyl derivatives, process for their preparation and pharmaceutical compositions containing them 法国施维雅药厂 2022-03-18 CN disclosed