SCHEMBL29639573

SCHEMBL29639573

COC(=O)NCc1ccccc1Br

nearest known ligand 0.58

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
RIPK1 Q13546 1/20 0.58
ALDH1A1 P00352 3/20 0.55
KMT2A Q03164 3/20 0.54
MEN1 O00255 1/20 0.50
NPC1 O15118 1/20 0.50
RAB9A P51151 1/20 0.50
ANPEP P15144 1/20 0.50
P2RX7 Q99572 4/20 0.48
KCNA5 P22460 1/20 0.47
LMNA P02545 1/20 0.47
MAPT P10636 1/20 0.47
EPHX2 P34913 1/20 0.46
HDAC1 Q13547 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9664850 0.87 KCNA5 (0.52) ALDH1A1KMT2AMEN1NPC1RAB9A
SCHEMBL1329466 0.83 RIPK1 (0.60) RIPK1ALDH1A1KMT2AMEN1NPC1
SCHEMBL12851863 0.83 TAAR1 (0.56) RIPK1KMT2ANPC1RAB9A
SCHEMBL102342 0.81 RIPK1 (0.61) RIPK1ALDH1A1KMT2AMEN1NPC1
SCHEMBL24242025 0.81 P2RX7 (0.54) RIPK1ALDH1A1KMT2AMEN1NPC1
SCHEMBL2749015 0.80 RIPK1 (0.52) RIPK1ALDH1A1KMT2AMEN1NPC1
SCHEMBL28333273 0.80 ALDH1A1 (0.62) ALDH1A1KMT2AMEN1NPC1RAB9A
SCHEMBL3416627 0.80 RIPK1 (0.52) RIPK1ALDH1A1KMT2ANPC1RAB9A
SCHEMBL2456852 0.79 KMT2A (0.58) RIPK1ALDH1A1KMT2AMEN1NPC1
SCHEMBL8583106 0.79 LMNA (0.55) RIPK1KMT2AKCNA5LMNAHDAC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3609905-B1 PEPTIDE MACROCYCLES AND USE THEREOF IN THE TREATMENT OF BACTERIAL INFECTIONS HOFFMANN LA ROCHE (CH) 2022-06-08 EP disclosed