SCHEMBL29640645

SCHEMBL29640645

COc1ccc(OCCC#N)cc1Br

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GAA P10253 2/20 0.44
KMT2A Q03164 1/20 0.43
L3MBTL1 Q9Y468 4/20 0.40
MAPT P10636 3/20 0.40
ALDH1A1 P00352 3/20 0.40
HPGD P15428 2/20 0.40
TDP1 Q9NUW8 2/20 0.40
SMN1; SMN2 Q16637 2/20 0.40
HSD17B10 Q99714 2/20 0.40
NPC1 O15118 1/20 0.40
RAB9A P51151 1/20 0.40
CASP1 P29466 1/20 0.40
MAPK1 P28482 2/20 0.38
LMNA P02545 1/20 0.38
AR P10275 1/20 0.38
PDE4A P27815 1/20 0.38
PDE4B Q07343 1/20 0.38
PDE4C Q08493 1/20 0.38
PDE4D Q08499 1/20 0.38
PPARD Q03181 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL23362964 1.00 GAA (0.44) GAAKMT2AL3MBTL1MAPTALDH1A1
SCHEMBL10746305 0.87 CA2 (0.52) GAAKMT2AALDH1A1HSD17B10CASP1
SCHEMBL2778087 0.84 GAA (0.44) GAAKMT2AL3MBTL1MAPTALDH1A1
SCHEMBL517916 0.80 L3MBTL1 (0.45) KMT2AL3MBTL1MAPTALDH1A1HPGD
SCHEMBL31648415 0.78 L3MBTL1 (0.46) L3MBTL1MAPTALDH1A1HPGDTDP1
SCHEMBL1810628 0.77 GAA (0.58) GAAKMT2AL3MBTL1MAPTALDH1A1
SCHEMBL28882436 0.75 ALDH1A1 (0.45) L3MBTL1MAPTALDH1A1HPGDTDP1
SCHEMBL16119617 0.75 HTR7 (0.51) MAPTALDH1A1LMNA
SCHEMBL10667947 0.75 MAPT (0.48) GAAKMT2AL3MBTL1MAPTALDH1A1
SCHEMBL9044971 0.75 MAPK1 (0.56) KMT2AL3MBTL1ALDH1A1TDP1HSD17B10

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-114641477-B Compounds having inhibitory activity on glucosylceramide synthase or pharmaceutically acceptable salts thereof and pharmaceutical compositions containing the same 柳韩洋行 2024-03-12 CN disclosed
CN-114641477-A Novel compound having inhibitory activity against glucose ceramide synthase or pharmaceutically acceptable salt thereof, method for preparing same, and pharmaceutical composition comprising same 柳韩洋行 2022-06-17 CN disclosed