SCHEMBL29643391

SCHEMBL29643391

COc1ccc(C#Cc2ccccc2)c([N+](=O)[O-])c1

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
RAB9A P51151 6/20 0.49
NPC1 O15118 4/20 0.49
SMN1; SMN2 Q16637 4/20 0.49
MAPT P10636 3/20 0.49
MAPK1 P28482 2/20 0.49
AKR1C3 P42330 4/20 0.47
AKR1C2 P52895 4/20 0.47
MMP2 P08253 1/20 0.46
MMP9 P14780 1/20 0.46
ALDH1A1 P00352 5/20 0.46
KMT2A Q03164 3/20 0.45
AKR1B10 O60218 2/20 0.44
AKR1B1 P15121 2/20 0.44
AKR1C4 P17516 2/20 0.44
AKR1C1 Q04828 2/20 0.44
MEN1 O00255 2/20 0.44
POLB P06746 2/20 0.44
KDM4E B2RXH2 1/20 0.43
CA12 O43570 1/20 0.42
CA1 P00915 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28641030 1.00 RAB9A (0.49) RAB9ANPC1SMN1; SMN2MAPTMAPK1
SCHEMBL28760471 0.89 AKR1C3 (0.47) RAB9ANPC1SMN1; SMN2MAPTMAPK1
SCHEMBL28484882 0.82 SMN1; SMN2 (0.54) RAB9ANPC1SMN1; SMN2MAPTMAPK1
SCHEMBL13931954 0.82 MAPK1 (0.46) RAB9ANPC1SMN1; SMN2MAPTMAPK1
SCHEMBL19063495 0.81 TSHR (0.51) RAB9ANPC1ALDH1A1CA12CA2
SCHEMBL29643377 0.81 TSHR (0.51) RAB9ANPC1ALDH1A1CA12CA2
SCHEMBL14387571 0.79 ALDH1A1 (0.42) RAB9ANPC1SMN1; SMN2MAPTMAPK1
SCHEMBL19622953 0.79 CASP3 (0.53) SMN1; SMN2MAPTMAPK1ALDH1A1KMT2A
SCHEMBL28041879 0.79 VCAM1 (0.52) SMN1; SMN2MAPTAKR1C3AKR1C2ALDH1A1
SCHEMBL4883148 0.78 ALDH1A1 (0.47) RAB9ANPC1SMN1; SMN2MAPTMAPK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-113429424-B Preparation method of [1,2,4] oxadiazino indoline-3-ketone derivative 华侨大学 2022-06-07 CN claimed
CN-113429424-B Preparation method of [1,2,4] oxadiazino indoline-3-ketone derivative 华侨大学 2022-06-07 CN disclosed