SCHEMBL29645433

SCHEMBL29645433

COc1ccc(-c2nc3c4cccc(Br)c4nc(Nc4ccccnc4=O)n3n2)c(C(F)(F)F)c1

nearest known ligand 0.33

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
P2RX7 Q99572 7/20 0.33
USP1 O94782 1/20 0.33
WDR48 Q8TAF3 1/20 0.33
THRB P10828 3/20 0.33
RXFP1 Q9HBX9 1/20 0.33
MAPK14 Q16539 1/20 0.33
GLO1 Q04760 1/20 0.33
KDM4E B2RXH2 1/20 0.33
ALDH1A1 P00352 1/20 0.33
POLB P06746 1/20 0.33
TP53 P04637 1/20 0.32
MAPT P10636 3/20 0.32
SMN1; SMN2 Q16637 1/20 0.32
CYP1A2 P05177 1/20 0.32
CYP3A4 P08684 1/20 0.32
ALOX15 P16050 1/20 0.32
TSHR P16473 1/20 0.32
CYP2C19 P33261 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29645580 0.90 P2RX7 (0.36) P2RX7THRBRXFP1KDM4EALDH1A1
SCHEMBL29645588 0.88 MAPT (0.43) P2RX7USP1WDR48THRBRXFP1
SCHEMBL29646008 0.84 KDM4E (0.47) THRBRXFP1KDM4EALDH1A1POLB
SCHEMBL29645803 0.83 POLB (0.46) P2RX7THRBRXFP1KDM4EALDH1A1
SCHEMBL29645431 0.81 SLC40A1 (0.35) P2RX7USP1WDR48POLB
SCHEMBL29645960 0.81 P2RX7 (0.33) P2RX7MAPT
SCHEMBL22980060 0.78 KDM4E (0.36) KDM4EALDH1A1
SCHEMBL22988389 0.78 KDM4E (0.36) KDM4EALDH1A1
SCHEMBL29645642 0.78 MAPT (0.43) P2RX7THRBRXFP1KDM4EPOLB
SCHEMBL29645475 0.77 KDM4E (0.44) THRBRXFP1KDM4EALDH1A1POLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-114466850-B [1,2,4] Triazolo [1,5-C ] quinazolin-5-amine 拜耳股份有限公司 2024-09-10 CN claimed
CN-114466850-A [1,2,4] triazolo [1,5-C ] quinazolin-5-amines 拜耳股份有限公司 2022-05-10 CN claimed