SCHEMBL29645592

SCHEMBL29645592

CCn1cc(-c2nc3c4cccc(C(F)(F)F)c4nc(Nc4ccccnc4=O)n3n2)c(C)n1

nearest known ligand 0.35

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
CYP1A2 P05177 1/20 0.35
LRRK2 Q5S007 1/20 0.35
P2RX7 Q99572 9/20 0.34
ADORA3 P0DMS8 5/20 0.33
ADORA2A P29274 5/20 0.33
ADORA1 P30542 5/20 0.33
ADORA2B P29275 4/20 0.33
KDM4E B2RXH2 2/20 0.33
ALDH1A1 P00352 1/20 0.33
HPGD P15428 1/20 0.33
TDP1 Q9NUW8 2/20 0.33
POLB P06746 1/20 0.33
THRB P10828 1/20 0.33
MAPT P10636 1/20 0.32
MEN1 O00255 1/20 0.31
CASP1 P29466 1/20 0.31
KMT2A Q03164 1/20 0.31
ESR2 Q92731 1/20 0.31
HSD17B10 Q99714 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL31150047 0.91 CYP1A2 (0.35) CYP1A2LRRK2P2RX7ADORA3ADORA2A
SCHEMBL29646056 0.89 ALDH1A1 (0.34) P2RX7ADORA3ADORA2AADORA1ADORA2B
SCHEMBL29646105 0.89 ADORA2A (0.38) P2RX7ADORA3ADORA2AADORA1ADORA2B
SCHEMBL29646061 0.88 KDM4E (0.34) P2RX7ADORA3ADORA2AADORA1ADORA2B
SCHEMBL29646221 0.88 CYP1A2 (0.35) CYP1A2LRRK2P2RX7MAPT
SCHEMBL29645615 0.87 ADORA3 (0.40) P2RX7ADORA3ADORA2AADORA1ADORA2B
SCHEMBL29645798 0.86 KDM4E (0.33) P2RX7ADORA3ADORA2AADORA1ADORA2B
SCHEMBL29646123 0.85 P2RX7 (0.33) P2RX7KDM4EALDH1A1HPGDTDP1
SCHEMBL29645597 0.83 TRPA1 (0.34) LRRK2P2RX7
SCHEMBL29646083 0.82 MAPT (0.35) P2RX7MAPTKMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-114466850-A [1,2,4] triazolo [1,5-C ] quinazolin-5-amines 拜耳股份有限公司 2022-05-10 CN claimed