SCHEMBL29645600

SCHEMBL29645600

CC(C)n1cc(-c2nc3c4cccc(C(F)(F)F)c4nc(Nc4ccccnc4=O)n3n2)cn1

nearest known ligand 0.33

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PDK2 Q15119 1/20 0.32
P2RX7 Q99572 5/20 0.32
ADORA3 P0DMS8 1/20 0.32
ADORA2A P29274 1/20 0.32
ADORA1 P30542 1/20 0.32
PDE3B Q13370 1/20 0.32
PDE3A Q14432 1/20 0.32
SLC40A1 Q9NP59 1/20 0.32
JAK2 O60674 2/20 0.31
ADA P00813 1/20 0.31
KDM5B Q9UGL1 1/20 0.31
PSEN1 P49768 1/20 0.31
PSEN2 P49810 1/20 0.31
APH1B Q8WW43 1/20 0.31
NCSTN Q92542 1/20 0.31
APH1A Q96BI3 1/20 0.31
PSENEN Q9NZ42 1/20 0.31
TYK2 P29597 1/20 0.31
HSP90AA1 P07900 1/20 0.30
AURKA O14965 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29645878 0.94 HSP90AA1 (0.35) P2RX7ADORA3ADORA2AADORA1PDE3B
SCHEMBL31149922 0.92 LIMK1 (0.35) ADORA3ADORA2AADORA1PDE3BPDE3A
SCHEMBL31150076 0.90 JAK2 (0.33) ADORA3ADORA2AADORA1JAK2KDM5B
SCHEMBL29645811 0.89 SLC40A1 (0.34) PDK2P2RX7SLC40A1JAK2AURKB
SCHEMBL29645797 0.88 JAK2 (0.32) P2RX7ADORA3ADORA2AADORA1JAK2
SCHEMBL29645601 0.88 MAPT (0.35) P2RX7ADORA3JAK2KDM5BTYK2
SCHEMBL29645561 0.87 MAP3K5 (0.34) P2RX7
SCHEMBL29646040 0.87 JAK2 (0.31) P2RX7JAK2KDM5BAURKALIMK1
SCHEMBL29645692 0.86 BRD4 (0.32) JAK2KDM5BTYK2AURKALIMK1
SCHEMBL29645717 0.85 FLT3 (0.32) PDK2JAK2KDM5BTYK2AURKB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-114466850-A [1,2,4] triazolo [1,5-C ] quinazolin-5-amines 拜耳股份有限公司 2022-05-10 CN claimed