SCHEMBL29645878

SCHEMBL29645878

O=c1nccccc1Nc1nc2c(C(F)(F)F)cccc2c2nc(-c3cnn(C(F)F)c3)nn12

nearest known ligand 0.35

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
HSP90AA1 P07900 3/20 0.35
TTK P33981 1/20 0.32
ADORA3 P0DMS8 1/20 0.32
ADORA2A P29274 1/20 0.32
ADORA1 P30542 1/20 0.32
P2RX7 Q99572 6/20 0.31
SLC40A1 Q9NP59 1/20 0.31
ADA P00813 1/20 0.31
PDE3B Q13370 3/20 0.31
PDE3A Q14432 3/20 0.31
PSEN1 P49768 1/20 0.30
PSEN2 P49810 1/20 0.30
APH1B Q8WW43 1/20 0.30
NCSTN Q92542 1/20 0.30
APH1A Q96BI3 1/20 0.30
PSENEN Q9NZ42 1/20 0.30
SCN9A Q15858 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29645600 0.94 PDK2 (0.32) HSP90AA1ADORA3ADORA2AADORA1P2RX7
SCHEMBL29645421 0.89 TTK (0.31) TTK
SCHEMBL31149922 0.86 LIMK1 (0.35) ADORA3ADORA2AADORA1PDE3BPDE3A
SCHEMBL29645561 0.86 MAP3K5 (0.34) P2RX7SCN9A
SCHEMBL29645537 0.86 MAPT (0.41) ADORA3ADORA1
SCHEMBL29645837 0.84 EGFR (0.36) P2RX7SLC40A1PSEN1PSEN2APH1B
SCHEMBL31150076 0.84 JAK2 (0.33) ADORA3ADORA2AADORA1
SCHEMBL29645682 0.84 ADORA3 (0.40) ADORA3ADORA2AADORA1P2RX7
SCHEMBL29645914 0.83 NR1H2 (0.40) ADORA3ADORA2AADORA1P2RX7
SCHEMBL29645601 0.83 MAPT (0.35) ADORA3P2RX7

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-114466850-A [1,2,4] triazolo [1,5-C ] quinazolin-5-amines 拜耳股份有限公司 2022-05-10 CN claimed