SCHEMBL29645825

SCHEMBL29645825

O=c1nccccc1Nc1nc2c(Br)cccc2c2nc(-c3ccc(F)cc3)nn12

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TP53 P04637 2/20 0.41
ADORA3 P0DMS8 9/20 0.39
ADORA1 P30542 4/20 0.39
ADORA2A P29274 5/20 0.37
MAPT P10636 2/20 0.37
XDH P47989 1/20 0.37
ABCG2 Q9UNQ0 1/20 0.34
RXFP1 Q9HBX9 2/20 0.34
GABRP O00591 1/20 0.34
GABRD O14764 1/20 0.34
GABRA1 P14867 1/20 0.34
GABRB1 P18505 1/20 0.34
GABRG2 P18507 1/20 0.34
GABRB3 P28472 1/20 0.34
GABRA5 P31644 1/20 0.34
GABRA3 P34903 1/20 0.34
GABRA2 P47869 1/20 0.34
GABRB2 P47870 1/20 0.34
GABRA4 P48169 1/20 0.34
GABRE P78334 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29645799 0.91 LMNA (0.38) TP53MAPTABCG2RXFP1
SCHEMBL29645755 0.91 MAPT (0.40) ADORA3ADORA1ADORA2AMAPTXDH
SCHEMBL29645618 0.90 ADORA3 (0.40) TP53ADORA3ADORA1ADORA2AMAPT
SCHEMBL29645930 0.90 POLB (0.38) TP53ADORA3ADORA1ADORA2AMAPT
SCHEMBL31149969 0.90 RXFP1 (0.38) TP53ADORA3ADORA1ADORA2AMAPT
SCHEMBL29645824 0.90 ADORA3 (0.39) TP53ADORA3ADORA1ADORA2AMAPT
SCHEMBL29645933 0.89 TP53 (0.41) TP53ADORA3ADORA1ADORA2AMAPT
SCHEMBL29646008 0.88 KDM4E (0.47) TP53ADORA3ADORA1ADORA2AMAPT
SCHEMBL29645976 0.87 KDM1A (0.36) TP53ADORA3ADORA2AMAPTRXFP1
SCHEMBL29645682 0.87 ADORA3 (0.40) TP53ADORA3ADORA1ADORA2AMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-114466850-A [1,2,4] triazolo [1,5-C ] quinazolin-5-amines 拜耳股份有限公司 2022-05-10 CN claimed