SCHEMBL29645682

SCHEMBL29645682

O=c1nccccc1Nc1nc2c(C(F)(F)F)cccc2c2nc(-c3ccc(F)cc3)nn12

nearest known ligand 0.40

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
ADORA3 P0DMS8 8/20 0.40
ADORA1 P30542 6/20 0.40
NR1H2 P55055 5/20 0.38
NR1H3 Q13133 5/20 0.38
ADORA2A P29274 4/20 0.38
NR1I2 O75469 1/20 0.38
NR3C1 P04150 1/20 0.38
MAPT P10636 1/20 0.38
TP53 P04637 2/20 0.38
P2RX7 Q99572 1/20 0.37
XDH P47989 1/20 0.36
SMN1; SMN2 Q16637 1/20 0.35
RXFP1 Q9HBX9 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29645914 0.92 NR1H2 (0.40) ADORA3ADORA1NR1H2NR1H3ADORA2A
SCHEMBL29646148 0.91 LMNA (0.39) MAPTTP53RXFP1
SCHEMBL29645803 0.90 POLB (0.46) ADORA3ADORA1ADORA2AMAPTTP53
SCHEMBL31149962 0.90 ADORA3 (0.39) ADORA3ADORA1NR1H2NR1H3ADORA2A
SCHEMBL29645618 0.89 ADORA3 (0.40) ADORA3ADORA1ADORA2AMAPTTP53
SCHEMBL29645933 0.87 TP53 (0.41) ADORA3ADORA1ADORA2AMAPTTP53
SCHEMBL29645825 0.87 TP53 (0.41) ADORA3ADORA1ADORA2AMAPTTP53
SCHEMBL29645837 0.86 EGFR (0.36) TP53P2RX7XDHSMN1; SMN2RXFP1
SCHEMBL29646027 0.85 MAPT (0.36) ADORA3ADORA1NR1H2NR1H3ADORA2A
SCHEMBL29645738 0.85 NTRK1 (0.36) ADORA3ADORA1ADORA2AP2RX7

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-114466850-A [1,2,4] triazolo [1,5-C ] quinazolin-5-amines 拜耳股份有限公司 2022-05-10 CN claimed