SCHEMBL29645908

SCHEMBL29645908

O=c1nccccc1Nc1nc2c(C(F)(F)F)cccc2c2nc(-c3cnn(CC4CCC4)c3)nn12

nearest known ligand 0.33

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
RIPK1 Q13546 1/20 0.33
EGFR P00533 1/20 0.33
CYP1A2 P05177 1/20 0.33
KCNH2 Q12809 1/20 0.33
GRM2 Q14416 1/20 0.33
PDK2 Q15119 2/20 0.32
CLK2 P49760 1/20 0.32
LRRK2 Q5S007 1/20 0.32
TBK1 Q9UHD2 5/20 0.32
ADORA3 P0DMS8 3/20 0.31
FLT3 P36888 1/20 0.31
IKBKE Q14164 1/20 0.31
STK17A Q9UEE5 1/20 0.31
RPS6KA6 Q9UK32 1/20 0.31
PIK3CA P42336 1/20 0.31
TTK P33981 1/20 0.31
SCN9A Q15858 1/20 0.31
GPR39 O43194 1/20 0.31
P2RX7 Q99572 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29645716 0.89 ADORA3 (0.32) EGFRKCNH2GRM2LRRK2TBK1
SCHEMBL29645561 0.87 MAP3K5 (0.34) PIK3CASCN9AP2RX7
SCHEMBL29645471 0.86 MAPT (0.40) EGFRADORA3
SCHEMBL29645916 0.86 EGFR (0.34) EGFRADORA3
SCHEMBL29645600 0.84 PDK2 (0.32) PDK2ADORA3P2RX7
SCHEMBL29645878 0.83 HSP90AA1 (0.35) ADORA3TTKSCN9AP2RX7
SCHEMBL29645998 0.83 MAPT (0.41) EGFRADORA3
SCHEMBL31149866 0.82 DYRK3 (0.35) CLK2ADORA3STK17APIK3CA
SCHEMBL31150114 0.81 ADORA3 (0.33) EGFRTBK1ADORA3TTK
SCHEMBL22980061 0.81 RIPK1 (0.34) RIPK1CYP1A2KCNH2GRM2PDK2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-114466850-A [1,2,4] triazolo [1,5-C ] quinazolin-5-amines 拜耳股份有限公司 2022-05-10 CN claimed