SCHEMBL29645922

SCHEMBL29645922

COc1ccc2nc(Nc3ccccnc3=O)n3nc(-c4cnn(C)c4)nc3c2c1

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ADORA3 P0DMS8 4/20 0.42
MAPT P10636 4/20 0.41
THRB P10828 2/20 0.41
RXFP1 Q9HBX9 2/20 0.41
POLB P06746 3/20 0.40
HPGD P15428 1/20 0.40
UBE2N P61088 1/20 0.40
TDP1 Q9NUW8 1/20 0.40
TP53 P04637 2/20 0.40
SMN1; SMN2 Q16637 2/20 0.39
CCNA2 P20248 2/20 0.39
CDK2 P24941 2/20 0.39
TTK P33981 2/20 0.39
KDM4E B2RXH2 2/20 0.38
ALDH1A1 P00352 1/20 0.38
FGFR2 P21802 1/20 0.38
KDR P35968 1/20 0.38
FGFR4 P22455 1/20 0.38
FGFR3 P22607 1/20 0.38
GAA P10253 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29645919 0.93 MAPT (0.41) ADORA3MAPTTHRBRXFP1POLB
SCHEMBL29646322 0.89 RXFP1 (0.40) ADORA3MAPTTHRBRXFP1TP53
SCHEMBL29645943 0.89 MAPT (0.50) ADORA3MAPTTHRBRXFP1POLB
SCHEMBL29645874 0.88 ADORA3 (0.40) ADORA3MAPT
SCHEMBL29645783 0.88 ADORA3 (0.42) ADORA3
SCHEMBL29645782 0.88 MAPT (0.43) ADORA3MAPTTHRBRXFP1POLB
SCHEMBL29646053 0.86 ADORA3 (0.41) ADORA3TTK
SCHEMBL29645577 0.85 MAPT (0.45) ADORA3MAPTTHRBRXFP1POLB
SCHEMBL29645835 0.83 ADORA3 (0.39) ADORA3MAPTRXFP1POLBALDH1A1
SCHEMBL29646002 0.83 MAPT (0.48) ADORA3MAPTTHRBRXFP1POLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-114466850-A [1,2,4] triazolo [1,5-C ] quinazolin-5-amines 拜耳股份有限公司 2022-05-10 CN claimed