SCHEMBL29660938

SCHEMBL29660938

NC(=O)c1ncccc1C1(C(F)(F)F)CC1

nearest known ligand 0.41

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
PDK2 Q15119 7/20 0.41
KDM4E B2RXH2 2/20 0.38
MAPT P10636 2/20 0.38
ALDH1A1 P00352 1/20 0.38
CYP3A4 P08684 1/20 0.38
ALOX15 P16050 1/20 0.38
TSHR P16473 1/20 0.38
BLM P54132 1/20 0.38
AGER Q15109 1/20 0.38
NPSR1 Q6W5P4 1/20 0.38
L3MBTL1 Q9Y468 1/20 0.38
RORC P51449 7/20 0.36
SMN1; SMN2 Q16637 1/20 0.34
CYP1A2 P05177 1/20 0.34
PARP1 P09874 1/20 0.34
P2RX7 Q99572 2/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29660959 0.87 PDK2 (0.38) PDK2KDM4EMAPTALDH1A1CYP3A4
SCHEMBL30829295 0.81 L3MBTL1 (0.48) PDK2KDM4EALDH1A1ALOX15L3MBTL1
SCHEMBL29661036 0.77 KDM4E (0.39) PDK2KDM4EMAPTALDH1A1CYP3A4
SCHEMBL30066845 0.76 KDM4E (0.41) KDM4EMAPTALDH1A1CYP3A4ALOX15
SCHEMBL31026277 0.76 PDK2 (0.42) PDK2KDM4EMAPTALDH1A1BLM
SCHEMBL22443382 0.74 PDK2 (0.51) PDK2KDM4EMAPTALDH1A1TSHR
SCHEMBL28911965 0.74 PARP1 (0.40) KDM4EMAPTALDH1A1CYP3A4ALOX15
SCHEMBL29660939 0.72 KDM4E (0.37) PDK2KDM4EMAPTALDH1A1CYP3A4
SCHEMBL29660941 0.72 SPR (0.37) KDM4EMAPTALDH1A1CYP3A4ALOX15
SCHEMBL18726259 0.71

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-117777126-A Imidazopyridines as IRAK4 degradants and uses thereof 武汉人福创新药物研发中心有限公司 2024-03-29 CN disclosed
EP-4003516-A1 PYRIDINE DERIVATIVES AS TMEM16A MODULATORS FOR USE IN THE TREATMENT OF RESPIRATORY CONDITIONS TMEM16A LIMITED (GB) 2022-06-01 EP disclosed