SCHEMBL2967281

SCHEMBL2967281

CNC(=O)COC(=O)NCCC1CCN(Cc2cccc(Cl)c2F)CC1

nearest known ligand 0.45

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
CHRM4 P08173 8/20 0.45
ACHE P22303 2/20 0.44
MAOA P21397 1/20 0.44
MAOB P27338 1/20 0.44
P2RX7 Q99572 1/20 0.42
FAAH O00519 1/20 0.42
CHRM2 P08172 2/20 0.42
TP53 P04637 1/20 0.41
ALPL P05186 1/20 0.41
ALPI P09923 1/20 0.41
ALPG P10696 1/20 0.41
CHRM5 P08912 1/20 0.41
CHRM1 P11229 1/20 0.41
CHRM3 P20309 1/20 0.41
KDM4E B2RXH2 1/20 0.41
POLB P06746 1/20 0.41
TSHR P16473 1/20 0.41
SMN1; SMN2 Q16637 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2972067 0.91 CXCR4 (0.49) CHRM4ACHEMAOAMAOBFAAH
SCHEMBL2974765 0.85 CHRM4 (0.45) CHRM4ACHEMAOAMAOBFAAH
SCHEMBL2967604 0.85 DRD2 (0.46) CHRM4ACHEMAOAMAOBP2RX7
SCHEMBL2977323 0.83 FAAH (0.48) CHRM4ACHEMAOAMAOBFAAH
SCHEMBL2979937 0.83 FAAH (0.48) CHRM4ACHEMAOAMAOBFAAH
SCHEMBL2981989 0.83 KCNH2 (0.46) CHRM4ACHEMAOAMAOBFAAH
SCHEMBL2979063 0.83 OPRM1 (0.51) CHRM4ACHE
SCHEMBL2974797 0.82 CHRM4 (0.49) CHRM4ACHEMAOAMAOBCHRM2
SCHEMBL3946467 0.82 ACHE (0.52) CHRM4ACHEMAOAMAOBCHRM2
SCHEMBL2974338 0.82 KDM4E (0.44) CHRM4ACHEFAAHTP53KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1720550-B1 DERIVATIVES OF PIPERIDINYLALKYLCARBAMATES, PREPARATION METHOD THEREOF AND USE OF SAME AS FAAH ENZYME INHIBITORS SANOFI AVENTIS (FR) 2009-04-15 EP claimed
US-20100279998-A1 PIPERIDINYLALKYLCARBAMATE DERIVATIVES, METHODS FOR THEIR PREPARATION AND THE THERAPEUTIC USE THEREOF AS FATTY ACID AMIDO HYDROLASE ENZYME INHIBITORS SANOFI-AVENTIS (FR) 2010-11-04 US disclosed
US-7781590-B2 Piperidinylalkylcarbamate derivatives, methods for their preparation and the therapeutic use thereof as fatty acid amido hydrolase enzyme inhibitors SANOFI-AVENTIS (FR) 2010-08-24 US disclosed
US-20070021403-A1 PIPERIDINYLALKYLCARBAMATE DERIVATIVES, METHODS FOR THEIR PREPARATION AND THE THERAPEUTIC USE THEREOF AS FATTY ACID AMIDO HYDROLASE ENZYME INHIBITORS SANOFI-AVENTIS (FR) 2007-01-25 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20100279998-A1 PIPERIDINYLALKYLCARBAMATE DERIVATIVES, METHODS FOR THEIR PREPARATION AND THE THERAPEUTIC USE THEREOF AS FATTY ACID AMIDO HYDROLASE ENZYME INHIBITORS FAAH, FAAH2, CNR2 CHRM4 2647/4885ACHE 428/4885MAOA 604/4885
US-20070021403-A1 PIPERIDINYLALKYLCARBAMATE DERIVATIVES, METHODS FOR THEIR PREPARATION AND THE THERAPEUTIC USE THEREOF AS FATTY ACID AMIDO HYDROLASE ENZYME INHIBITORS FAAH, FAAH2, CNR2 CHRM4 2788/4885ACHE 455/4885MAOA 635/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.