SCHEMBL29699673

SCHEMBL29699673

O=C(NO)c1cccc(CN2C(=O)C(=O)c3ccccc32)c1

nearest known ligand 0.59

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CES1 P23141 4/20 0.59
ALDH1A1 P00352 4/20 0.59
CHRM1 P11229 2/20 0.59
ALDH2 P05091 2/20 0.59
ALDH3A1 P30838 2/20 0.59
HPGD P15428 1/20 0.56
HTT P42858 1/20 0.56
CHRM5 P08912 2/20 0.54
CHRM3 P20309 1/20 0.54
ACHE P22303 2/20 0.54
BCHE P06276 2/20 0.54
APAF1 O14727 1/20 0.54
TP53 P04637 1/20 0.54
CYP1A2 P05177 1/20 0.54
CYP3A4 P08684 1/20 0.54
CYP2D6 P10635 1/20 0.54
MAPT P10636 1/20 0.54
ALOX15 P16050 1/20 0.54
TSHR P16473 1/20 0.54
ALOX12 P18054 1/20 0.54

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28468478 1.00 CES1 (0.59) CES1ALDH1A1CHRM1ALDH2ALDH3A1
SCHEMBL28799632 0.87 ALDH1A1 (0.65) CES1ALDH1A1CHRM1ALDH2ALDH3A1
SCHEMBL28799598 0.86 ALDH3A1 (0.65) CES1ALDH1A1ALDH2ALDH3A1ACHE
SCHEMBL28467222 0.86 CTRB1 (0.48) ALDH1A1ALDH2ALDH3A1ACHEHDAC1
SCHEMBL18954771 0.86 KMT2A (0.72) CES1ALDH1A1CHRM1ALDH2ALDH3A1
SCHEMBL28462499 0.86 HDAC1 (0.72) CES1ALDH1A1CHRM1ALDH2ALDH3A1
SCHEMBL281838 0.84 TRPA1 (0.71) CES1ALDH1A1CHRM1ALDH2ALDH3A1
SCHEMBL29699601 0.82 CASP1 (0.67) ALDH1A1ALDH2ALDH3A1HPGDHTT
SCHEMBL28799595 0.82 CASP1 (0.67) ALDH1A1ALDH2ALDH3A1HPGDHTT
SCHEMBL18974295 0.79 CHRM1 (0.71) CES1ALDH1A1CHRM1ALDH2ALDH3A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-111747883-B 1-benzyl isatin derivative and synthesis method and application thereof 中南大学 2022-07-01 CN disclosed