SCHEMBL29742908

SCHEMBL29742908

O=C(O)c1csc(-c2cccc(OC(F)(F)F)c2)c1

nearest known ligand 0.50

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
LDHA P00338 1/20 0.50
HSD17B1 P14061 1/20 0.48
HSD17B2 P37059 1/20 0.48
DHODH Q02127 8/20 0.47
CSNK2A2 P19784 1/20 0.46
CSNK2B P67870 1/20 0.46
CTSA P10619 1/20 0.45
STK17B O94768 1/20 0.44
MRGPRX4 Q96LA9 1/20 0.44
AURKA O14965 1/20 0.44
TPX2 Q9ULW0 1/20 0.44
ABL1 P00519 1/20 0.43
SLC13A5 Q86YT5 1/20 0.43
IGF2BP2 Q9Y6M1 1/20 0.43
RXRA P19793 1/20 0.43
RXRB P28702 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28923987 1.00 LDHA (0.50) LDHAHSD17B1HSD17B2DHODHCSNK2A2
SCHEMBL29742864 0.86 RXRA (0.49) LDHAHSD17B1HSD17B2MRGPRX4RXRA
SCHEMBL28634234 0.86 RXRA (0.49) LDHAHSD17B1HSD17B2MRGPRX4RXRA
SCHEMBL29742784 0.83 HSD17B1 (0.67) HSD17B1HSD17B2RXRARXRB
SCHEMBL28635415 0.83 HSD17B1 (0.67) HSD17B1HSD17B2RXRARXRB
SCHEMBL5515377 0.81 KMO (0.56) DHODHCSNK2A2CSNK2BMRGPRX4AURKA
SCHEMBL938500 0.80 KMO (0.52) HSD17B1HSD17B2DHODH
SCHEMBL505417 0.80 RXRA (0.61) DHODHCSNK2A2CSNK2BAURKATPX2
SCHEMBL29784241 0.80 RXRA (0.61) DHODHCSNK2A2CSNK2BAURKATPX2
SCHEMBL24952187 0.78 ALDH1A1 (0.57) LDHARXRARXRB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-113444081-B Thiadiazole carboxamide compounds and application thereof 浙江大学 2022-07-05 CN disclosed