SCHEMBL2975469

SCHEMBL2975469

COc1c(Nc2cccc3[nH]ccc23)cccc1OCCCl

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
RET P07949 1/20 0.47
HTR1B P28222 1/20 0.45
JAK2 O60674 1/20 0.43
JAK3 P52333 1/20 0.43
HTR1A P08908 4/20 0.42
MAPK14 Q16539 1/20 0.42
PRKCQ Q04759 1/20 0.41
DRD2 P14416 1/20 0.41
DRD4 P21917 1/20 0.41
DRD3 P35462 1/20 0.41
SRC P12931 1/20 0.41
MEN1 O00255 1/20 0.39
MAPT P10636 1/20 0.39
MAPK1 P28482 1/20 0.39
KMT2A Q03164 1/20 0.39
PIK3CD O00329 1/20 0.39
PIK3CA P42336 1/20 0.39
PIK3CB P42338 1/20 0.39
MTOR P42345 1/20 0.39
PIK3CG P48736 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2986267 0.86 RET (0.45) RETHTR1BJAK2JAK3HTR1A
SCHEMBL2982161 0.85 RET (0.54) RETHTR1BJAK2JAK3MAPK14
SCHEMBL17255752 0.83 TSHR (0.51) RETHTR1BHTR1ADRD2DRD4
SCHEMBL17255754 0.81 SRC (0.46) RETHTR1BJAK2JAK3HTR1A
SCHEMBL2980702 0.80 ULK1 (0.45) RETJAK2MAPK14PRKCQTUBB4A
SCHEMBL17255769 0.80 PRKCQ (0.46) RETHTR1BJAK2JAK3MAPK14
SCHEMBL4073823 0.77 HTR1B (0.60) HTR1BHTR1ADRD2DRD4DRD3
SCHEMBL1545429 0.72 HTR1B (0.60) HTR1BHTR1ADRD2DRD4DRD3
SCHEMBL7876385 0.70 HTR1B (0.58) HTR1BHTR1ADRD2DRD4DRD3
SCHEMBL9130728 0.70 HDAC3 (0.52) MEN1MAPTMAPK1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7781591-B2 Substituted 3-cyanopyridines as protein kinase inhibitors WYETH LLC (US) 2010-08-24 US claimed