SCHEMBL2986267

SCHEMBL2986267

COc1c(Nc2cccc3[nH]ccc23)cccc1OCCN(C)C

nearest known ligand 0.45

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
RET P07949 1/20 0.45
HTR7 P34969 2/20 0.44
HTR1B P28222 2/20 0.44
HTR1A P08908 4/20 0.42
JAK2 O60674 1/20 0.41
JAK3 P52333 1/20 0.41
ALDH1A1 P00352 1/20 0.41
MAPK14 Q16539 1/20 0.41
PRKCQ Q04759 1/20 0.40
DRD2 P14416 1/20 0.40
DRD4 P21917 1/20 0.40
DRD3 P35462 1/20 0.40
SRC P12931 1/20 0.40
NR4A2 P43354 2/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2975469 0.86 RET (0.47) RETHTR1BHTR1AJAK2JAK3
SCHEMBL2982161 0.83 RET (0.54) RETHTR1BJAK2JAK3MAPK14
SCHEMBL17255752 0.81 TSHR (0.51) RETHTR1BHTR1AALDH1A1DRD2
SCHEMBL2980622 0.81 NR4A2 (0.46) HTR7HTR1BJAK2ALDH1A1PRKCQ
SCHEMBL4864576 0.80 HTR1A (0.60) HTR7HTR1BHTR1AALDH1A1DRD2
SCHEMBL17255754 0.77 SRC (0.46) RETHTR1BHTR1AJAK2JAK3
SCHEMBL9132797 0.77 RXFP1 (0.58) ALDH1A1NR4A2
SCHEMBL9130935 0.73 NR4A2 (0.53) HTR1ANR4A2
SCHEMBL10736779 0.72 HTR1B (0.49) HTR7HTR1BHTR1ADRD2DRD4
SCHEMBL10736784 0.72 HTR1B (0.49) HTR7HTR1BHTR1ADRD2DRD4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7781591-B2 Substituted 3-cyanopyridines as protein kinase inhibitors WYETH LLC (US) 2010-08-24 US claimed