SCHEMBL2977948

SCHEMBL2977948

COCc1ccc2c(c1)ncn2-c1cccc(COCc2nccn2C)c1

nearest known ligand 0.39

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
FGFR1 P11362 11/20 0.39
KIT P10721 1/20 0.37
FLT3 P36888 1/20 0.37
KDR P35968 1/20 0.36
GABRA1 P14867 1/20 0.35
GABRG2 P18507 1/20 0.35
GABRB3 P28472 1/20 0.35
GABRA5 P31644 1/20 0.35
GABRA3 P34903 1/20 0.35
GABRA2 P47869 1/20 0.35
SRC P12931 2/20 0.35
HPGD P15428 3/20 0.35
ALDH1A1 P00352 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2974096 0.91 FGFR1 (0.38) FGFR1KITFLT3GABRA1GABRG2
SCHEMBL13202763 0.91 PRKCI (0.40) FGFR1KITFLT3GABRA1GABRG2
SCHEMBL2652208 0.87 SIGMAR1 (0.43) FGFR1KDRSRCHPGDALDH1A1
SCHEMBL2966387 0.85 KMT2A (0.48) FGFR1GABRA1GABRG2GABRB3GABRA5
SCHEMBL2978335 0.85 NPC1 (0.40) FGFR1KITFLT3HPGD
SCHEMBL2966791 0.84 FGFR1 (0.39) FGFR1KITFLT3KDRSRC
SCHEMBL13202762 0.84 APP (0.34) FGFR1KITFLT3GABRA1GABRG2
SCHEMBL2652697 0.83 KMT2A (0.37) FGFR1GABRA1GABRG2GABRB3GABRA5
SCHEMBL2652685 0.82 GABRA1 (0.47) FGFR1KITFLT3KDRGABRA1
SCHEMBL2653362 0.82 FGFR1 (0.39) FGFR1KITFLT3KDRGABRA1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7776900-B2 Benzimidazole derivatives and their use for modulating the GABAAreceptor complex NEUROSEARCH A/S (DK) 2010-08-17 US claimed
US-20090030018-A1 Benzimidazole derivatives and their use for modulating the gabaalpha receptor complex ANIONA APS (DK) 2009-01-29 US claimed
US-7776900-B2 Benzimidazole derivatives and their use for modulating the GABAAreceptor complex NEUROSEARCH A/S (DK) 2010-08-17 US disclosed
US-20090030018-A1 Benzimidazole derivatives and their use for modulating the gabaalpha receptor complex ANIONA APS (DK) 2009-01-29 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20090030018-A1 Benzimidazole derivatives and their use for modulating the gabaalpha receptor complex GABRB2, GABRB1, GABRB3 FGFR1 4324/4885KIT 3187/4885FLT3 2451/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.